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3-(2-methylphenyl)-N-(4H-1,2,4-triazol-4-yl)propanamide
3-[2-(3-fluorophenyl)ethyl]-1-(1H-imidazol-4-ylmethyl)piperidine
1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-4-[2-(pyridin-2-yl)ethyl]piperazine
{[(3S,4R)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
1-cyclohexanecarbonyl-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-N-methylpyrrolidine-2-carboxamide
6-methoxy-1-[(4-methoxyphenyl)methyl]-4-[2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]-1,4-diazepan-2-one
3-{1-[(4-ethylphenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)acetamide
ethyl 4-(3-methyl-1-propyl-1H-pyrazole-4-amido)piperidine-1-carboxylate
1-(carbamoylmethyl)-N-[(2-ethoxypyridin-3-yl)methyl]piperidine-3-carboxamide
2-ethyl-1-[(1-ethylpyrrolidin-2-yl)methyl]-6-methyl-4-oxo-N-{[3-(trifluoromethyl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
6-[(2-methylphenyl)methyl]-N-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
5-acetyl-N-methyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
3-methyl-5-(phenoxymethyl)-N-[1-(1,3-thiazol-2-yl)ethyl]furan-2-carboxamide
4-(2-{3-[3-(6-methoxypyridin-2-yl)phenyl]-1H-pyrazol-1-yl}ethyl)morpholine
1-[2-(morpholin-4-yl)ethyl]-6-oxo-N-[(1-phenylcyclohexyl)methyl]piperidine-3-carboxamide
ethyl 1-[(2-chlorophenyl)methyl]-4-(cyclopropylmethyl)piperidine-4-carboxylate
4-[(1-benzyl-1H-imidazol-2-yl)methyl]-2-(trifluoromethyl)morpholine
7-(1-benzoxepine-4-carbonyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)oxolane-3-carboxamide
(2R,6R)-4-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2R,4S)-4-hydroxy-1-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperidine-2-carboxylic acid
3-{2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
4-({2-[2-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}methyl)quinoline
5-chloro-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[(2,4-dimethoxy-3-methylphenyl)methyl]-N-(pyridin-3-ylmethyl)piperazine-2-carboxamide
5-[3-(pyridine-2-carbonyl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
(2S,3R)-2-amino-3-hydroxy-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
4-[(4-fluorophenyl)methyl]-1-(1-methylpiperidin-4-yl)-3-(propan-2-yl)-1,4-diazepan-5-one
3-ethyl-N-(1H-indol-3-yl)-5-methyl-1,2-oxazole-4-carboxamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-(2-methoxyethyl)-N-(propan-2-yl)benzamide
2-[(4-chlorophenyl)methyl]-8-{spiro[2.3]hexane-1-carbonyl}-2,8-diazaspiro[4.5]decan-3-one
3-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
3-(3-methyl-1H-pyrazol-1-yl)-1-[9-(oxan-2-ylmethoxy)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
3-(1-benzofuran-2-yl)-4-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}-1H-pyrazole
2-(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)ethan-1-ol
methyl 4-[({2-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]ethyl}amino)methyl]benzoate
2-methoxy-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]quinoline-4-carboxamide
ethyl 1-(pyridin-2-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2-methylpropanamide
(3aS,6aS)-2-(2-aminopyrimidin-4-yl)-5-cyclopentyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}-1-(3-sulfamoylphenyl)urea
ethyl 3-benzyl-1-(1H-imidazol-2-ylmethyl)piperidine-3-carboxylate
2-{4-[(2-methoxyphenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
5-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]-1,2-oxazol-3-ol
8-(5-chloro-7-methoxy-1-benzofuran-2-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
4-(4-{2-[1-(propan-2-yl)piperidin-4-yl]acetyl}piperazin-1-yl)benzonitrile
2-(2-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)ethan-1-ol