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(1H-imidazol-2-ylmethyl)(methyl){[4-(5-methylfuran-2-yl)phenyl]methyl}amine
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-4-(3-fluorophenyl)benzamide
2-{1-benzyl-4-[1-(4-chlorophenyl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-1H-1,3-benzodiazol-2-yl)methanol
N-ethyl-2-[4-methyl-6-(morpholine-4-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-yl]-N-(propan-2-yl)acetamide
1-methyl-5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-1,3-benzodiazole
N-[1-(2-fluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-[2-(3-chlorophenyl)ethyl]-2-(methoxymethyl)-6-methyl-4-oxo-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1,4-dihydropyridine-3-carboxamide
1-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyridin-3-ylmethyl)piperazine
3-butyl-4-(2,3-dimethoxybenzoyl)-1-methylpiperazin-2-one
8-(1-benzothiophen-2-ylmethyl)-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]oxy}pyridine
(2R,3S,6R)-5-(2-ethylpyrimidine-5-carbonyl)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-1,3-oxazolidin-2-one
3,4,5-trimethoxy-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
1-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-3-ethoxypropan-1-one
1-(2-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
2-[4-(1H-1,3-benzodiazol-2-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-benzyl-2-methyl-5-(2-methylpropanamido)-N-(prop-2-en-1-yl)-1H-1,3-benzodiazole-7-carboxamide
N-methyl-2-({5-[(quinolin-6-yloxy)methyl]-1,2-oxazol-3-yl}formamido)acetamide
2-(3-chloro-4-hydroxyphenyl)-1-[2-(4-chlorophenyl)morpholin-4-yl]ethan-1-one
2-chloro-3-({[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)-9-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
9-[(3-fluoro-4-methoxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(5-methoxy-1,2-dimethyl-1H-indole-3-carbonyl)azetidin-3-ol
4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-1-methyl-1,4,9-triazaspiro[5.5]undecane
N-[3-(4-{[(1-benzyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]pyridine-3-carboxamide
2,3-dimethyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]quinoxaline-6-carboxamide
(3S,9aR)-3-(4-aminobutyl)-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[(2,6-difluorophenyl)methyl]-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-chloro-4-fluoro-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1-benzothiophene-2-carboxamide
N,5-dimethyl-N-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(4-methoxypyridin-2-yl)methyl]pyrrolidin-3-yl]cyclobutanecarboxamide
methyl 5-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-methyl-8-(6-methylpyridine-3-carbonyl)-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-{4-[1-(2,3-dimethylphenyl)piperidin-4-yl]piperazin-1-yl}-1-azabicyclo[2.2.2]octane
3-ethyl-N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-4,5-dihydro-1,2-oxazole-5-carboxamide
{1-[(3,5-dimethyl-1H-indol-2-yl)methyl]-4-(oxan-2-ylmethyl)piperidin-4-yl}methanol
4-methyl-6-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-2-amine
(2E)-N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)-3-(thiophen-2-yl)prop-2-enamide
2-[3-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)propyl]-1,3-benzothiazole
2-amino-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-6-(pyridin-2-yl)pyridine-3-carbonitrile
5-ethyl-5-(1-{[3-(2-hydroxyethoxy)phenyl]methyl}piperidin-4-yl)-3-[2-(4-methoxyphenyl)ethyl]imidazolidine-2,4-dione
5-{[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}-2-methoxyphenol
methyl 3-(oxolane-3-amido)-1-(3-phenylpropyl)-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
ethyl 4-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine-1-carboxylate
7-(5-chloropyridin-2-yl)-9-methoxy-4-[(4-methoxy-3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}pyridine
1-[(4-methoxyphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)benzoyl]piperazin-2-one
4-({1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-2-yl}methyl)morpholine