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3-chloro-N-[2-(4-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}phenoxy)propyl]benzamide
(4S)-1-(6-cyclopropylpyrimidin-4-yl)-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
2-{2-[1-(4-oxo-4H-chromene-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-[3-(cyclohexyloxy)propyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
(1R,3S)-3-amino-N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}cyclohexane-1-carboxamide
N-[3-(dimethylcarbamoyl)-5-({[1-(4-methoxyphenyl)propan-2-yl]amino}methyl)phenyl]pyridine-2-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(pyrimidin-2-ylmethyl)piperidin-4-yl]propanamide
2-(adamantan-1-yl)-1-[3-(piperidin-1-yl)azetidin-1-yl]ethan-1-one
4-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-5-methyl-1,3-oxazole
1-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-4-(1H-1,2,4-triazol-3-yl)benzamide
N-[3-(dimethylamino)propyl]-N-methyl-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-amine
5-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
4-[1-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazol-2-yl]-2-(propan-2-yl)pyrimidine
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidine
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
1-cycloheptyl-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)piperidin-2-one
1-[benzyl(methyl)amino]-3-[4-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]propan-2-ol
5-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
N-methyl-N-{[5-oxo-4-(2-phenoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-3-yl]methyl}methanesulfonamide
3-({[2-(3-methoxyphenyl)phenyl]carbamoyl}(methyl)amino)-N-methylbutanamide
1-(2-methoxyphenyl)-4-(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)piperazine
2-(4-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amino]methyl}phenoxy)ethan-1-ol
4-{1-[1-(3-chloro-5-methoxybenzoyl)piperidin-4-yl]ethyl}morpholine
1-{4-hydroxy-4-[2-(4-phenylazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-1-yl}-2-methoxyethan-1-one
1-[2-(benzyloxy)ethyl]-4-phenoxypiperidine-4-carboxylic acid
methyl[2-(1H-pyrazol-1-yl)ethyl]{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
1-(5-{[(2,1,3-benzoxadiazol-5-ylmethyl)amino]methyl}-2-methoxyphenoxy)-3-(piperidin-1-yl)propan-2-ol
(1R,5S,8R)-3-{[4-(5-methylfuran-2-yl)phenyl]methyl}-3-azabicyclo[3.2.1]octan-8-ol
3-[4-(furan-2-yl)butan-2-yl]-1-(6-methylpyridin-3-yl)urea
1-ethyl-N-[(1-hydroxycyclohexyl)methyl]-1H-indole-5-carboxamide
6-(2-chlorophenyl)-N-ethyl-N-(pyridin-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-{4-[(2,2-dimethylpyrrolidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}-1-[(2E)-2-methylpent-2-en-1-yl]piperidine
(1S,5R)-1,3,3-trimethyl-6-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-6-azabicyclo[3.2.1]octane
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-ethyl-8-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)benzonitrile
5-(1,4-dioxan-2-yl)-1-(4-fluorophenyl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazole
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamide
5-(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
1-methyl-4-[(5-{[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]methyl}-1,2,4-oxadiazol-3-yl)methyl]piperidine
N-(1H-1,3-benzodiazol-2-yl)-2-[(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)amino]acetamide
2-{5-[1-(1-methoxypropan-2-yl)-1H-imidazol-2-yl]furan-2-yl}-1-methyl-1H-1,3-benzodiazole
N-(cyclopropylmethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-N-propyl-1H-pyrazole-4-carboxamide
2-[2-(1-methylpiperidin-2-yl)ethyl]-1,2-dihydroisoquinolin-1-one
5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-(2-phenylethyl)piperidin-2-one
5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-3-(thiophen-2-yl)-1,2,4-oxadiazole
5-(3,4-dimethylphenoxymethyl)-N-[(1-ethylpyrrolidin-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]-1-[3-(1H-imidazol-5-yl)phenyl]urea