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N-[(4-tert-butyl-1,3-thiazol-2-yl)methyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-methoxy-3-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrazine
6-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-2-phenylimidazo[1,2-a]pyridine
N-[2-(2,3-dimethoxyphenyl)ethyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-ethyl-1-[2-(3-propanamidophenoxy)acetyl]pyrrolidine-3-carboxamide
2-[(4aR,7aS)-4-[2-(3-hydroxyphenyl)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
1-methyl-3-(4-{4-[(thiolan-3-yl)amino]piperidin-1-yl}phenyl)imidazolidin-2-one
methyl 3-acetamido-1-methyl-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
ethyl 1-[(3,5-dimethoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
2-(dimethylamino)-8-[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-(3-ethoxypropanoyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
4-(2-methoxyacetyl)-N-[2-(trifluoromethoxy)phenyl]-1,4-diazepane-1-carboxamide
N-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N-cyclopropylfuran-2-carboxamide
4-[(2-fluorophenyl)methyl]-1-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperidine
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(5-methyl-1H-pyrazol-1-yl)propanamide
4-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
(2S)-N-[2-(4-methoxyphenyl)phenyl]-1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidine-2-carboxamide
6-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]pyrazine-2-carboxamide
2-(2-cyclopropylpyrimidin-5-yl)-4-(3,3-dimethylpyrrolidine-1-carbonyl)-7-methylquinoline
methyl 5-[(oxan-4-yl)amino]-3-(oxolane-3-amido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(1-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}ethyl)morpholine
(2S,4S)-4-amino-N-[1-(benzenesulfonyl)piperidin-4-yl]-1-methylpyrrolidine-2-carboxamide
3-[1-(1,3-benzothiazole-5-carbonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2R)-2-amino-1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-hydroxypropan-1-one
2-cyclopropyl-8-[4-(4-methoxyphenyl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one
5-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-{5-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
3-{[1-propyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-3,4-dihydroquinazolin-4-one
{1-[(2,5-dimethylphenyl)methyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
methyl 1-{2-[1-(2H-1,3-benzodioxol-5-ylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetyl}piperidine-4-carboxylate
4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-ethyl-2-[(isoquinolin-5-yloxy)methyl]-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
5-{1-[(4-chlorophenyl)methyl]-3-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-ethyl-1H-imidazole
5-tert-butyl-4-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}furan-2-carboxamide
N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-[3-(azocane-1-carbonyl)piperidin-1-yl]-7-methanesulfonyl-4-methylquinazoline
1,1-dioxo-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
(1S,5R)-6-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-3-methyl-3,6-diazabicyclo[3.2.2]nonane
3-phenoxy-N-{1-[1-(2-phenylethyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[3-(pyridin-3-yloxy)propyl]amine
3-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
2-amino-4-(4-cyanophenyl)-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
7-(5-chloropyridin-2-yl)-4-(1,3-oxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{1-[({[3-fluoro-5-(trifluoromethyl)phenyl]methyl}carbamoyl)methyl]-1H-pyrazol-4-yl}-3-(2-methoxyphenyl)propanamide
N,N-diethyl-1-({4-[(3-fluoro-4-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-3-carboxamide
N-{2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]ethyl}pyridine-3-carboxamide