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2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]acetamide
7-(5-chloropyridin-2-yl)-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-benzyl-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
2-(3-hydroxypiperidin-1-yl)-N-methyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]acetamide
1-[(2-aminopyridin-3-yl)methyl]-4-(1H-pyrrole-2-carbonyl)-1,4-diazepan-6-ol
4'-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(1-ethylcyclobutyl)methyl]-4-{[(3R,4R)-4-hydroxypyrrolidin-3-yl]sulfamoyl}benzamide
2-(3-acetyl-1H-indol-1-yl)-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]acetamide
1-(2-{3-methyl-2-oxo-1-oxa-3,7-diazaspiro[4.5]decan-7-yl}-2-oxoethyl)-1H-indole-3-carboxamide
2-[({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)amino]pyridine-4-carboxamide
2-methyl-1-[1-(2-propyl-1,3-thiazole-4-carbonyl)azetidin-3-yl]piperidine
N-cyclopropyl-2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-4-carboxamide
2-(4-methoxy-2,6-dimethylphenyl)-2-[4-(2-methoxyethyl)piperazin-1-yl]acetic acid
N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-3-(1H-imidazol-4-yl)-2-(1H-pyrrol-1-yl)propanamide
3-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
4-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenol
N-[4-methoxy-3-({[4-(morpholin-4-yl)butan-2-yl]carbamoyl}amino)phenyl]acetamide
3-ethynyl-N-(2-hydroxyethyl)-N-(propan-2-yl)benzamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyrrolidine-1-sulfonamide
2-(4-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-1-yl)-1,3-benzothiazole
N-methyl-1-[(4-methylphenyl)amino]-N-(piperidin-3-ylmethyl)cyclopentane-1-carboxamide
N-methyl-5-[(quinolin-8-yloxy)methyl]-N-(thiophen-3-ylmethyl)-1,2-oxazole-3-carboxamide
1-[(2S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
N-{[5-(ethylsulfanyl)-1,3,4-oxadiazol-2-yl]methyl}-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
6-methyl-3-({4-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-{4-oxo-3H,4H-thieno[3,2-d]pyrimidin-3-yl}acetamide
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(methoxymethyl)piperidine
3-[(cyclopropylmethyl)amino]-N-[2-(1H-imidazol-1-yl)ethyl]-5-(phenylsulfamoyl)benzamide
2-[5-(methoxymethyl)furan-2-carbonyl]-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
2-{2-[1-(4-methylpiperazine-1-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
(1-{3-[(3-methoxyphenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidin-4-yl)diphenylmethanol
9-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
2-(4-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-1-(thiophen-2-ylmethyl)piperazin-2-yl)ethan-1-ol
(3R,4R)-4-ethyl-1-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)piperidine-3,4-diol
3-(dimethyl-1,2-oxazol-4-yl)-1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}propan-1-one
1-[6-hydroxy-4-(5-methyl-1,2,4-oxadiazol-3-yl)-1,4-diazepan-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
7-chloro-3-[(4-ethylpiperazin-1-yl)methyl]-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
(1R,7S)-3-(2-methoxyethyl)-N-methyl-4-oxo-N-(pyrazin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-[2-(4-phenylpiperidin-1-yl)ethyl]-3-propyl-1H-pyrazole-5-carboxamide
1-[(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)pyrrolidin-1-yl]-2-(2-ethyl-1H-imidazol-1-yl)ethan-1-one
5-(azepane-1-carbonyl)-N-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
2-ethyl-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N,4-dimethyl-1,3-oxazole-5-carboxamide
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
1-{[3-(4-benzylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-3-ol
N-(5-tert-butyl-2-methoxyphenyl)-2-(2-methoxyethyl)piperidine-1-carboxamide
2-[5-(2-amino-6-methoxypyrimidin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol