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4-[2-(2,1,3-benzoxadiazol-4-yl)-1H-imidazol-1-yl]benzene-1-sulfonamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
3-methyl-1-(2-methylpropyl)-8-[(3-phenoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3-methoxyphenyl)methyl]-4-(6-oxo-1,6-dihydropyridine-3-carbonyl)piperazin-2-one
N-[1-(1-cyclopropylethyl)-3-methyl-1H-pyrazol-5-yl]-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carboxamide
1-(2-chlorophenyl)-3-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(2-phenylethyl)acetamide
3-(3,4-dimethoxyphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
methyl 6-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-cyclopropanecarbonyl-8-(3-hydroxy-2-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[(3-cyclohexyl-1H-pyrazol-4-yl)methyl](methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
methyl[3-(1-methyl-1H-pyrazol-4-yl)propyl]{[(1R,5S,6R)-3-(2-methylbenzoyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}amine
3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1-methyl-1,2,5,6,7,8-hexahydroquinolin-2-one
6-fluoro-2-({[3-(1H-1,2,3-triazol-1-yl)propyl]amino}methyl)quinolin-4-ol
2-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-1H-1,3-benzodiazole
N-cyclopropyl-4-(4-methoxy-2-methylphenyl)benzamide
5-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]pyridine-2-carbonitrile
5-benzyl-5-{1-[3-(furan-2-yl)propanoyl]piperidin-4-yl}-3-[2-(pyrrolidin-1-yl)ethyl]imidazolidine-2,4-dione
1-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-3-[2-(2-methyl-4-phenylpiperazin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
methyl 2-[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]pyridine-3-carboxylate
N-[(6-methylpyridin-2-yl)methyl]-6-(naphthalene-1-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[1-(2-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)-1H-pyrazol-4-yl]pyridine-2-carboxamide
2-(2H-1,3-benzodioxol-5-yloxy)-1-[4-hydroxy-4-(hydroxymethyl)azepan-1-yl]ethan-1-one
4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1λ6-thiane-1,1-dione
1-(2-methoxyphenyl)-4-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1H-pyrazole
2-{[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]methyl}-1-methyl-1H-1,3-benzodiazole
3-{[3-(2-hydroxyethyl)-4-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-1-yl]methyl}phenol
ethyl 1-(5-methoxyfuran-2-carbonyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)[1-(1H-1,2,4-triazol-5-yl)ethyl]amine
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-4,6-dihydroxypyridine-3-carboxamide
ethyl 1-{1-[2-(cyclohexylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carbonyl}piperidine-4-carboxylate
(1R,2R,6S,7S)-4-[2,2-dimethyl-1-(3-methylthiophen-2-yl)cyclopropanecarbonyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
N-({5-[(2-butyl-1H-imidazol-4-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-[(1R,5R)-6-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-[(3,4-difluorophenyl)methyl]-5-[4-(2-ethoxyphenyl)piperazin-1-yl]azepan-2-one
N-{3-[4-(3-methoxyphenyl)-2-methyl-5-oxopiperazin-1-yl]-3-oxopropyl}methanesulfonamide
2-[1-benzyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(cyclopropylmethyl)-N-(oxolan-2-ylmethyl)acetamide
2-(4-acetylphenoxy)-1-{2-[2-(1H-imidazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
N-{1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}pyridin-2-amine
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(2-oxo-1,2-dihydropyridin-1-yl)acetamide
(1R,5R)-3-[3-(4-ethylphenyl)-1H-pyrazole-5-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
9-[(4-ethoxyphenyl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-phenoxyethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
1-[1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)benzamide
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-4-methoxybenzene-1-sulfonamide
3-(oxolan-2-yl)-7-{[4-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine