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2-[3-(3-fluorophenoxymethyl)-5-[(methylamino)(phenyl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
[1-(2-amino-5-ethyl-6-methylpyrimidin-4-yl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
2-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
5-{1-[(2E)-2-methylbut-2-enoyl]piperidin-4-yl}-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
8-(2,6-dimethylpyrimidine-4-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-[(2S)-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]pyrrolidine-2-carbonyl]morpholine
(2,3-dihydro-1-benzofuran-2-ylmethyl)({[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl})methylamine
2-[(1-cyclopentylpiperidin-4-yl)oxy]-5-methoxy-N-(1-phenylcyclopropyl)benzamide
2-{4-[2-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
ethyl 3-[(2-fluorophenyl)methyl]-1-(pyridine-2-carbonyl)piperidine-3-carboxylate
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-(quinolin-5-ylmethyl)pyrrolidin-3-yl]methanol
ethyl 1-[1-(4-{[(2-fluorophenyl)methyl]carbamoyl}phenyl)piperidin-4-yl]piperidine-4-carboxylate
2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(2R)-pyrrolidin-2-ylmethyl]acetamide
6-[(4-methoxynaphthalen-1-yl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
5-cyclobutanecarbonyl-3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-(4-ethylphenyl)-6-methylpyrimidin-2-amine
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
2-{2-[1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
1-(4-fluorophenyl)-4-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperazine
3-methyl-2-[(1S)-1-{5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}ethyl]pyridine
4-benzyl-3-ethyl-1-{[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
N-[2-(dimethylamino)ethyl]-2-fluoro-N-{[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl}benzamide
1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
N-[(3R,4S)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
1-[(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-3-yl)methyl]pyrrolidin-2-one
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-3-(4H-1,2,4-triazol-4-yl)benzamide
4-(2-{8-methyl-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
2-(2,4-dichlorophenoxy)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]acetamide
2-(methylamino)-N-[2-(4-methylbenzenesulfonyl)ethyl]pyridine-4-carboxamide
{6-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidine-1-carbonyl]pyridin-2-yl}methanol
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-(1-phenylethyl)benzamide
1-(azocan-1-yl)-3-(2-{[bis(2-hydroxyethyl)amino]methyl}-5-methoxyphenoxy)propan-2-ol
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-methyl-6-propylpyrimidin-4-amine
methyl 4-{4-[(1R,2R,3S,4S)-3-aminobicyclo[2.2.1]heptane-2-carbonyl]piperazin-1-yl}benzoate
3-(1H-1,3-benzodiazol-2-ylmethyl)-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
1-{[1-(cyclohexylmethyl)-2-cyclopropylmethanesulfonyl-1H-imidazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
1-cyclohexyl-N-methyl-N-[2-(4-methylphenoxy)ethyl]-1H-1,2,3-triazole-4-carboxamide
N,4-dimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,3-thiazol-2-amine
2-ethyl-6-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
3-[2-(2,3-dimethylphenoxy)ethyl]-1,3-diazinane-2,4-dione
6-[2-(4-chlorophenyl)morpholin-4-yl]-N-ethyl-N-methylpyrimidin-4-amine
4-benzoyl-1-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine
3-[(2-methoxyethyl)sulfamoyl]-5-(1H-1,2,3-triazol-1-yl)benzoic acid
methyl 2-(5-methyl-2-{[(2E)-3-(pyridin-2-yl)prop-2-enamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
5-{[4-(oxan-4-yl)piperazin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
(5S,9aS,9bS)-2-cyclopentyl-5-(2,5-dimethylphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]imidazo[1,2-a]pyridine-6-carboxamide
{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})amine
N-(2-hydroxyethyl)-N-(propan-2-yl)-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-{[2-(2-fluorophenyl)acetamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide