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methyl 5-{[(2,4-dimethoxy-3-methylphenyl)methyl]amino}-3-acetamido-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(2-benzylphenyl)-2-(2-methoxyethyl)morpholine-4-carboxamide
3-(4-methoxyphenyl)-N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazole-5-carboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(morpholin-4-yl)propyl]acetamide
N-[2-(1H-indol-1-yl)ethyl]-2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamide
4-(cyclopropylmethyl)-1-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-{[1-(dimethylamino)cyclohexyl]methyl}-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
3-(azetidine-1-carbonyl)-N-{[1-(ethoxymethyl)cyclobutyl]methyl}benzene-1-sulfonamide
2-acetyl-8-(4-aminopyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[2-(dimethylsulfamoyl)ethyl]-5-methyl-2-phenyl-1H-imidazole-4-carboxamide
2-[(2-chlorophenyl)methyl]-4-[4-(2-ethylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-benzyl-8-(1H-indol-3-ylmethyl)-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
(1S,5R)-3-(1H-imidazol-2-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-3-(1-methylpiperidin-2-yl)propanamide
N-benzyl-N-(cyclopropylmethyl)-3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
4-(2-methoxyphenoxy)-1-(2-methyl-5-propylpyrimidin-4-yl)piperidine-4-carboxylic acid
1-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
ethyl 1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-3-(3-phenylpropyl)piperidine-3-carboxylate
N-benzyl-3-({[(2,4-difluorophenyl)methyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
{1-[(2,5-dimethoxyphenyl)methyl]-4-(2-phenylethyl)piperidin-4-yl}methanol
N-({4-[(2-chloroprop-2-en-1-yl)oxy]phenyl}methyl)-2-fluoro-N-(pyridin-3-ylmethyl)benzamide
6-[(diethylamino)methyl]-N-(2,2-difluoroethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(2-chloro-5-sulfamoylphenyl)azocane-1-carboxamide
2-[3-(furan-2-yl)-5-[2-(5-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-1H-1,2,4-triazol-1-yl]acetic acid
2-hydroxy-N-[(3R,4S)-4-propyl-1-[(trimethyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]acetamide
1-[2-(2H-1,3-benzodioxol-5-yl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
5-{3-[4-(3-chlorophenoxy)piperidin-1-yl]-3-oxopropyl}-5-[(4-fluoro-3-methoxyphenyl)methyl]pyrrolidin-2-one
3-{[(1-{[3-(difluoromethoxy)phenyl]methyl}piperidin-4-yl)oxy]methyl}pyridine
ethyl 1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-[4-(3-methoxyphenyl)piperazin-1-yl]-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]ethan-1-one
1-ethyl-2-{1-[(2-methoxyphenyl)methyl]-1H-imidazol-2-yl}-1H-imidazole
9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-(naphthalen-1-ylmethyl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
8-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]acetyl}-2,8-diazaspiro[4.5]decan-3-one
4-(5-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidine-1-carbonyl}pyridin-2-yl)piperazin-2-one
15-methyl-12-(4-methylpiperazine-1-carbonyl)-9-(3-methylthiophen-2-yl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-3-(methanesulfonylmethyl)piperidine
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-(3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanoyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
4-[6-(pyrimidin-5-yl)pyridazin-3-yl]thiomorpholine
1-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethan-1-one
2-methyl-3-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-benzyl-5-{[3-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}pyrimidin-2-amine
1-{4-[2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]phenyl}imidazolidine-2,4-dione
N-[(5-benzyl-1,2,4-oxadiazol-3-yl)methyl]-1-propanoylpiperidine-3-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amine
1-(propane-2-sulfonyl)-3-[3-(trifluoromethyl)benzoyl]piperidine
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-acetamido-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
7-(1,3-benzothiazol-2-yl)-4-(2,2-difluoroethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol