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5-fluoro-2-[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
(2R,6R)-2,6-bis(prop-2-en-1-yl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}-1,2,3,6-tetrahydropyridine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1-phenylcyclopropane-1-carboxamide
2-[4-({methyl[1-(pyridin-2-yl)propan-2-yl]amino}methyl)phenoxy]-1-(pyrrolidin-1-yl)ethan-1-one
3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)-5-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-cyclopropyl-3-{1-[2-(phenylsulfanyl)acetyl]piperidin-3-yl}propanamide
N-[4-(4-{[(2,6-difluoro-3-methylphenyl)methyl]amino}piperidin-1-yl)phenyl]-2-fluorobenzamide
N-methyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
7-{[3-(2-aminoethyl)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetamide
2-[benzyl({[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
4-[3-(morpholin-4-ylmethyl)phenyl]pyridin-3-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-methylacetamide
1-{[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]amino}propan-2-ol
(3S,4S)-1-(4-methyl-1,3-thiazole-5-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
3-(3-methylbutyl)-8-(2-propyl-1,3-thiazole-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1,9-dioxaspiro[5.5]undecan-4-amine
(4aS,8aR)-1-(3-methylbutyl)-6-(6-oxo-1,6-dihydropyridazine-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
ethyl 2-{4-[1-(6-ethoxy-4-methylquinazolin-2-yl)piperidin-4-yl]morpholin-3-yl}acetate
N,N-dimethyl-7-(1-methylcyclopropanecarbonyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[2-(1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidin-2-yl)ethyl]phenol
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-propylfuran-2-yl)methyl]piperidine
3-({4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
[(2E)-3-(furan-2-yl)prop-2-en-1-yl][3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amine
[5-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxypropyl)piperidine
(3R,4R)-1-(4-chloro-3-fluorobenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
1-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-cyclohexylpiperazine
1-cyclohexyl-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-[3-(1,3-oxazol-5-yl)phenyl]urea
N-(2,3-dihydro-1H-inden-1-yl)-4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
6-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-2-methoxy-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
2-{[(3S)-1-benzylpiperidin-3-yl]amino}-N-(pyrazin-2-yl)acetamide
2-(benzyloxy)-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
2-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}-N-(2-methoxy-5-methylphenyl)acetamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(4,4,4-trifluorobutanoyl)-decahydro-1,6-naphthyridin-2-one
5-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4-ethyl-1,3-thiazol-2-amine
(2S,4R)-4-amino-N-methyl-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidine-2-carboxamide
3-{2,7-diazaspiro[4.5]decane-7-carbonyl}-4-phenyl-1H-pyrazol-5-amine
N-[(4-methylphenyl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
ethyl 4-(2-phenoxyethyl)-1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxylate
N-(4-fluoro-2-methylphenyl)-3-{1-[3-(pyridin-3-yl)propanoyl]piperidin-3-yl}propanamide
methyl 2-[7-chloro-3-({[2-(diethylamino)ethyl](ethyl)amino}methyl)-2-oxo-1,2-dihydroquinolin-1-yl]acetate
(2S,4R)-1-(1-benzothiophene-2-carbonyl)-4-(dimethylamino)pyrrolidine-2-carboxylic acid
4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-(4-{4-[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)amino]piperidin-1-yl}phenyl)-2-phenoxyacetamide
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(ethyl)(pyridin-4-ylmethyl)amine
(3S,4S)-1-(4-aminopyridine-2-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
2-({[(3R,4R)-1-[1-(3,5-dimethylphenyl)piperidin-4-yl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
N-({6-[4-(hydroxymethyl)phenyl]pyridin-3-yl}methyl)acetamide
2-phenyl-N-[(7-{[3-(trifluoromethyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide