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3-{5-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
5-{2-[2-(ethylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}quinoline
1-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(3-methoxyphenyl)propan-1-one
3-chloro-N-cyclopentyl-4-{[1-(2-oxopropanoyl)piperidin-4-yl]oxy}benzamide
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-[2-(2-methoxyethyl)piperidin-1-yl]propan-1-one
(3S,4R)-1-(2H-1,3-benzodioxole-5-carbonyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
1-ethyl-4-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine
5-(2,4-dimethoxyphenyl)-N-[2-phenyl-2-(piperidin-1-yl)ethyl]-1,2,4-triazin-3-amine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[3-(hydroxymethyl)pyrrolidin-1-yl]pyridine-3-carboxamide
5-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-3-(phenoxymethyl)-1,2,4-oxadiazole
(4aS,8aR)-1-(3-methylbutyl)-6-[3-(pyrazin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
3-(4-methoxyphenyl)-1-{4-[2-(oxolan-2-yl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}propan-1-one
[1,4-bis({[3-(trifluoromethyl)phenyl]methyl})piperidin-4-yl]methanol
[1-(2,3-dihydro-1H-inden-2-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]methanol
5-(2,6-difluorophenoxymethyl)-N-{[3-(methylsulfanyl)phenyl]methyl}-1,2-oxazole-3-carboxamide
1-{2-cyclopentyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-3-(methoxymethyl)pyrrolidine
2-{2-[1-(2H-1,3-benzodioxol-5-yl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]ethyl}-1-methylpiperidine
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxy-N-methyl-N-(oxan-2-ylmethyl)benzamide
5-(2-methyl-1,3-benzothiazol-5-yl)-1,2,3,4-tetrahydroisoquinoline
1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
N-(1-{2-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2H-1,3-benzodioxole-5-carboxamide
2-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}morpholin-3-yl)acetic acid
4-[(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)carbamoyl]pyridin-1-ium-1-olate
N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}oxane-4-carboxamide
(1R,2S,9R)-11-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-3-(thiophen-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N,N-dimethyl-2-(1-{[3-(2-methylpropyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}cyclopentyl)acetamide
{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(piperidin-3-ylmethyl)amine
1-cyclopropyl-4-[4-(3-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]pyrrolidin-2-one
methyl 1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine-2-carboxylate
4-(4-{[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]amino}piperidin-1-yl)-N-[2-(morpholin-4-yl)ethyl]benzamide
4-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-3-fluoropyridine
2-{4-[2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]piperazin-1-yl}ethan-1-ol
2-(2-chloroprop-2-en-1-yl)-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
4,6-dimethyl-3-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
7-(5-methylthiophen-2-yl)-4-[(2S)-piperidine-2-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2,2-dimethyloxan-4-yl)-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-(2-{7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
1'-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-(6-hydroxy-1,4-oxazepan-4-yl)-1-(1,2,3,4-tetrahydroquinolin-1-yl)propan-1-one
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)oxane-2-carboxamide
7-[3-(pyridin-2-yl)propanoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
4-ethyl-N-[4-(3-methoxyphenoxy)phenyl]-2-methyl-3-oxopiperazine-1-carboxamide
5-benzyl-4-cyclobutanecarbonyl-1-(4-methylphenyl)piperazin-2-one
(2S,4R)-1-[(4-chlorophenyl)methyl]-N,N-diethyl-4-[(1-propylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide
N-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-4-fluoro-3-methylbenzene-1-sulfonamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-propyl-1H-pyrazole-5-carboxamide
5-[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]-2-methyl-2,3-dihydropyridazin-3-one