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N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-(4-fluorophenyl)-4-(4-methyl-1,3-thiazol-2-yl)-1,4-diazepane
5-[4-(3-hydroxy-3-methylbutyl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
1-(2-fluorophenyl)-N-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-ethyl-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
4-benzyl-3-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[4-methoxy-3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)cyclohexanecarboxamide
3,5-dichloro-N-(1,1-dioxo-1λ6-thian-4-yl)-N,4-dimethylbenzamide
1-(4-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-[3-(dimethylcarbamoyl)propanoyl]-N-[4-(2-fluorophenoxy)phenyl]piperidine-2-carboxamide
[2-(azepan-1-yl)ethyl](ethyl){[5-(oxan-2-yl)furan-2-yl]methyl}amine
ethyl 4-[3-(ethylcarbamoyl)pyridin-2-yl]piperazine-1-carboxylate
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-[(3-methylpyridin-4-yl)methyl]pyridin-2-amine
1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
2-oxo-8-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-[1-(pyridin-2-yl)piperidine-3-carbonyl]-1,4-diazepan-2-one
(4aR,7aS)-1-cyclopropanecarbonyl-4-(5-methoxyfuran-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(2,5-dimethylphenyl)-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
4-(4-{[2-(hydroxymethyl)phenyl]methyl}piperazine-1-carbonyl)benzonitrile
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N,1-dimethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
5-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)propanamide
3-butanamido-N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]benzamide
3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-methyl-2-(4-methylphenoxymethyl)-1-(pyridin-2-ylmethyl)-1,4-dihydropyridin-4-one
1-cyclopropyl-3-(4-methoxyphenyl)-3-(2-{4-[(2-methylphenyl)methyl]piperazin-1-yl}-2-oxoethyl)pyrrolidine-2,5-dione
N-({7-[(2-hydroxy-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methylbutanamide
3-({[(2-aminopyridin-3-yl)methyl]amino}methyl)-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
(5S,9aS,9bS)-2-cyclopentyl-5-(2-fluoro-5-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-chloro-1-methyl-N-{1-[(2-methylphenyl)methyl]cyclopropyl}-1H-pyrazole-5-carboxamide
1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(2-methylphenoxy)piperidine
N-(3-methoxypropyl)-N-(1-methylpiperidin-4-yl)-1-[2-(naphthalen-1-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
3-(1H-imidazol-2-yl)-N-methyl-N-(quinolin-5-ylmethyl)benzamide
1-ethyl-3-(pyridin-2-ylmethyl)-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-methylthiophene-2-carboxamide
1-(2-ethoxyethyl)-N-methyl-2-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
methyl({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})[2-(pyridin-2-yl)ethyl]amine
3-(4-benzyl-1H-pyrazol-5-yl)-1-{imidazo[1,2-a]pyridine-3-carbonyl}piperidine
8-[3-(1,3-benzothiazol-2-yl)propanoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(4aS,8aR)-6-(4-methyl-1H-imidazole-5-carbonyl)-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
methyl 4-{[(2-{1-[2-(3-methoxyphenyl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
6-methyl-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-[(2R,3R)-1'-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
7-(1-benzothiophen-3-yl)-9-ethoxy-4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-{[3-(4-ethylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}quinoline
5-(2-fluorophenyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-amino-1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-[2-(1H-imidazol-4-yl)ethyl]-2-methyl-3-[(pyridin-3-ylmethyl)amino]benzamide
6-[({[4-(1H-pyrazol-1-yl)phenyl]methyl}amino)methyl]-1,4-oxazepan-6-ol