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5-(1-{[3-(benzyloxy)phenyl]methyl}piperidin-4-yl)-5-(2-phenylethyl)imidazolidine-2,4-dione
2-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-2,3-dihydro-1,2-benzothiazol-3-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
1-(cyclopropylmethyl)-N-ethyl-5-[2-(2H-indazol-2-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[1-(3,5-dichloro-4-methylphenyl)-N-methylformamido]-N-methylbutanamide
3-ethyl-1-[4-(3-methoxyphenoxy)phenyl]-3-(oxan-2-ylmethyl)urea
(4aR,7aS)-1-methyl-4-(2-phenoxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3-methoxyphenyl)methyl]-3-(4-methylpiperazin-1-yl)-N-(prop-2-en-1-yl)propanamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(thiophen-3-yl)acetamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-(4-methoxybenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[3-(dimethylamino)propyl]piperidine-3,5-dicarboxamide
3-[(3-cyanopiperidin-1-yl)sulfonyl]-N-[3-(methylsulfanyl)propyl]benzamide
2-(1-benzylpiperidin-4-yl)-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]ethan-1-one
N-(butan-2-yl)-N-(thiophen-3-ylmethyl)-1H-1,2,3-benzotriazole-5-carboxamide
2-methyl-5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-1H-1,3-benzodiazole
1-{2-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-2-oxoethyl}-1,4-dihydroquinolin-4-one
2-(2,5-difluorophenyl)-1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]ethan-1-one
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
N-[2-(2-hydroxyethoxy)ethyl]-2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)acetamide
3-{2-[2-(pyridin-3-yl)morpholin-4-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N,3,5,7-tetramethyl-N-[(2-methylpyridin-4-yl)methyl]-1H-indole-2-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-(4-methoxyphenyl)-4-{1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}piperazine
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethylimidazo[2,1-b][1,3]thiazole-6-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
1-[2-(1-{2-[3-(trifluoromethyl)phenyl]acetyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
6-(2-methylphenyl)-N-(quinolin-6-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-({2-[(2-oxopyrrolidin-1-yl)methyl]phenyl}methyl)-4-(piperidin-3-yl)benzamide
N-methyl-N-(oxan-4-yl)-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
N-(dimethyl-1H-1,2,4-triazol-5-yl)-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
2-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)quinolin-8-ol
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
ethyl 4-[3-(carbamoylmethyl)-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl]piperidine-1-carboxylate
2-(adamantan-1-yl)-5-(azepane-1-carbonyl)pyrimidin-4-ol
5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(4aR,8aS)-6-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-1-[(3,4,5-trimethoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
dimethyl({4-methyl-5-[1-(9H-purin-6-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
{[4-(cyclopentyloxy)phenyl]methyl}({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
3-(1H-imidazol-1-ylmethyl)-1-[(2,3,4-trifluorophenyl)methyl]piperidine
1-cyclopropyl-3-{2-[2-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(4-methoxyphenyl)pyrrolidine-2,5-dione
2-[1-(3-phenoxybenzenesulfonyl)azetidin-3-yl]pyridine
(1S,6R)-3-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
2-amino-4-(2,6-dimethylphenyl)-6-(pyrazine-2-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-1,3-thiazole-4-carboxamide
1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
[(4-ethyl-5-{1-[(3-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
4-[(4-{2-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-2-yl]ethoxy}phenyl)methyl]piperazine-1-carbaldehyde
3-{4-[3-(1H-pyrazol-5-yl)phenyl]-1H-pyrazol-1-yl}propanamide