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5-[(2,4-dimethyl-1H-imidazol-1-yl)methyl]-3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazole
N'-(2,4-dimethylphenyl)-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}propanediamide
2-{2-[6-amino-5-cyano-4-(2,4-difluorophenyl)pyridin-2-yl]phenoxy}acetamide
methyl 1-ethoxy-2-oxo-8-[2-(pyridin-2-ylsulfanyl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-methyl-5-phenyl-1-[(1s,4s)-4-aminocyclohexyl]piperidin-2-one
N-[3-(3-methylphenyl)propyl]-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[(3-chlorophenyl)methyl]-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl]methanol
1-[(5-cyclopentylthiophen-2-yl)methyl]-3-(4H-1,2,4-triazol-3-yl)piperidine
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[(6-methylpyridin-2-yl)methyl]-1,2-oxazole-3-carboxamide
3-hydroxy-1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
5-(4-fluorophenyl)-7-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}pyrazolo[1,5-a]pyrimidine
4-(1-{1-[(4-fluoro-2-methylphenyl)methyl]piperidin-4-yl}ethyl)morpholine
1-{3-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}-2-(methoxymethyl)piperidine
2-chloro-6-methoxy-4-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenol
5-(methoxymethyl)-N-({3-methyl-7-[2-(2,3,6-trifluorophenyl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
5-{[3-(2-ethyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-oxazol-5-yl]methoxy}-2-methyl-1,3-benzothiazole
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-2-(5-methyl-1H-pyrazol-1-yl)acetamide
2-(adamantan-1-yl)-1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]ethan-1-one
ethyl 2-(1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
ethyl[2-(1H-pyrazol-1-yl)ethyl]{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}amine
9-[(2-methylpyrimidin-5-yl)methyl]-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}propanamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(3-methoxy-4-methylphenyl)propan-1-one
3-(2-{[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-1-hydroxyethyl)phenol
N-[(3-methoxyphenyl)methyl]-3-[1-(pyrimidin-2-yl)piperidin-3-yl]propanamide
3-[(3-fluorophenyl)methyl]-N-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-5-carboxamide
N-{1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyridin-2-amine
1-(2-{[(2,3-dichloro-4-methylphenyl)methyl](methyl)amino}ethyl)piperidin-2-one
4-{1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-2-methylpropan-2-yl}morpholine
1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methoxyethan-1-one
4-(5-fluoro-2-methylbenzenesulfonyl)-9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
9-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-3-azaspiro[5.5]undecane
5-(4-fluorophenyl)-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-1-methyl-1H-imidazole-2-carboxamide
N-{[7-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,2,5-thiadiazole-3-carboxamide
1-(2-cyclopropylacetyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-{3-[2-(pyridin-2-yl)-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
N-(3-hydroxy-2,2-dimethylpropyl)-2-(3-methoxyphenyl)-1,3-benzoxazole-6-carboxamide
1-(benzyloxy)-8-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzothiazole
4-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)carbamoyl)amino]-3-methyl-N-(propan-2-yl)benzamide
4-(4-ethoxyphenyl)-1-ethyl-3-methyl-1H-pyrazole
2-methyl-N-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl}methyl)benzene-1-sulfonamide
5,6-dimethyl-2-{2-oxo-2-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}-2,3-dihydropyridazin-3-one
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-4,5,6,7-tetrahydro-1,2-benzoxazole