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N-(1-benzothiophen-2-ylmethyl)-1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
3-(furan-2-ylmethyl)-5-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}-5-propylimidazolidine-2,4-dione
N-(1-methanesulfonylpiperidin-4-yl)-3-(1,2-oxazinan-2-yl)propanamide
3-methyl-N-[1-(1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]butanamide
[1-(7-chloro-2-methylquinoline-4-carbonyl)piperidin-2-yl]methanamine
4-[(4-fluorophenyl)methyl]-1-(5-fluoropyridine-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-{1-[7-(2H-1,3-benzodioxol-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-3-phenylpropanamide
2-{2-oxo-2-[4-(thian-4-yl)piperazin-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]propan-1-one
2-(3-methyl-1H-pyrazol-1-yl)-1-[4-(3-phenylpropyl)-1,4-diazepan-1-yl]ethan-1-one
1-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}-1H-1,2,4-triazole
(1R,5R)-6-[(2-butyl-1H-imidazol-4-yl)methyl]-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-{3-oxo-3-[3-(4-phenoxybenzoyl)piperidin-1-yl]propyl}piperidin-2-one
N-(2-cyano-3-methylphenyl)-4-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)benzamide
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
3-cyclopropaneamido-N-[2-(3,4-dimethylphenoxy)ethyl]-4-methylbenzamide
methyl({[1-(morpholin-4-yl)cyclohexyl]methyl})({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
1-(3-methylbutyl)-3-(pyridin-3-ylmethyl)-8-(1,3-thiazol-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-(oxolan-2-yl)-2-(3-{[(prop-2-en-1-yl)(pyridin-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-methyl-3-{1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(3-chlorophenyl)-N-cyclobutyl-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-[5-(4-chlorophenyl)-1H-pyrrol-2-yl]-1-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}propan-1-one
N-methyl-N-(1-methylpiperidin-4-yl)-3-{1-[(3,4,5-trimethoxyphenyl)methyl]piperidin-3-yl}propanamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
[(3R,5S)-5-(hydroxymethyl)-1-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperidin-3-yl]methanol
1-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}azetidin-3-yl)-3,5-dimethyl-1H-pyrazole
N-benzyl-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine-1-sulfonamide
4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(2-cyclopropylpyrimidin-5-yl)-N,N-diethyl-7,8-dimethylquinoline-4-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
5-chloro-6-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carboxylic acid
6-{4-[3-(pyridin-2-yl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}pyridine-3-carbonitrile
2-({4-[2-(dimethylamino)acetyl]-6-hydroxy-1,4-diazepan-1-yl}methyl)benzonitrile
1-[2-(4-ethyl-3,3-dimethylpiperazin-1-yl)-2-oxoethyl]-3-methoxy-1,2-dihydropyridin-2-one
6-[4-({2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}amino)piperidin-1-yl]pyridine-3-carbonitrile
4-hydroxy-N-methyl-2-(pyridin-3-yl)-N-[1-(pyrimidin-4-yl)ethyl]pyrimidine-5-carboxamide
3-methyl-7-[(2,3,4-trimethoxyphenyl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-[2-(1H-imidazol-4-yl)ethyl]propanamide
N-[(4-methoxyphenyl)methyl]-5-(2-methylbutanoyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(7-chloroquinolin-4-yl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3-[(5-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}furan-2-yl)sulfanyl]-4-methyl-4H-1,2,4-triazole
1-cycloheptyl-4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidine
[(3R,4R)-1-[(3-methylphenyl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
7-fluoro-3-methyl-N-[1-(thiophen-2-yl)propyl]-1-benzofuran-2-carboxamide
3-(3,4-dimethoxybenzoyl)-1-[(5-ethylthiophen-2-yl)sulfonyl]piperidine
5-methyl-1'-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]-2-(2-hydroxyphenyl)ethan-1-one
N-(1-methanesulfonylpiperidin-4-yl)-5-(oxolan-2-yl)thiophene-2-carboxamide
N,N-diethyl-2-[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetamide
(2S,4S)-N-methyl-1-(propan-2-yl)-4-{[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]amino}pyrrolidine-2-carboxamide