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N-[(6-chloropyridin-3-yl)methyl]-N-methyl-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
6-(2-chloro-6-fluorophenyl)-N,N-dimethylpyridine-3-carboxamide
4-{4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}-1-[(2-chlorophenyl)methyl]piperidine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}propanamide
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
8-(4-phenyl-1H-imidazole-5-carbonyl)-1-oxa-8-azaspiro[4.5]decane
6-methyl-2-(4-methylphenoxymethyl)-1-[2-(morpholin-4-yl)ethyl]-3-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
N-{[3-(benzyloxy)phenyl]methyl}oxane-2-carboxamide
4-chloro-2-{[3-(2-hydroxyethyl)-4-(thiophen-3-ylmethyl)piperazin-1-yl]methyl}phenol
1-[(3-methoxyphenyl)methyl]-5-[(propan-2-yloxy)methyl]-1H-1,2,4-triazole
methyl 2-(azocane-1-sulfonyl)-6-cyclopentanecarbonyl-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
2-(1,3-benzothiazol-2-ylmethyl)-4-[3-(thiomorpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
(8aS)-2-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2,6-difluoro-N-[(7-{[4-(trifluoromethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-(1,3-thiazol-5-ylmethyl)-decahydro-2,7-naphthyridin-4a-ol
[(2-fluoro-4-methoxyphenyl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
[(5-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
8-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-(azepan-1-ylmethyl)-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-[(2-chlorophenyl)methyl]-3-{1-[4-(methylsulfanyl)benzoyl]piperidin-3-yl}propanamide
5-ethanesulfonamido-N,1-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-phenyl-1H-1,3-benzodiazole-7-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-{2-[(3,4-dimethoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
1-(2-methoxyphenyl)-4-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1H-pyrazole
N5-ethyl-N3-methyl-4-oxo-1-(2-phenylethyl)-N3-(quinolin-5-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
5-[1-ethyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
methyl (2S,4S)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(pyridine-2-amido)pyrrolidine-2-carboxylate
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-3-methyl-3H-[1,2,3]triazolo[4,5-b]pyridine-6-carboxamide
N'-[(4-chlorophenyl)methyl]-N'-(3-hydroxypropyl)-N-(2-methylphenyl)propanediamide
2-(adamantan-1-yl)-5-(4-methyl-1,4-diazepane-1-carbonyl)pyrimidin-4-ol
N,N-dimethyl-3-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]aniline
8-chloro-N-ethyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}quinoline-2-carboxamide
methyl (2S,4R)-1-(1-ethylpiperidin-4-yl)-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
2-[1-(6-methoxy-3-methyl-1-benzofuran-2-yl)-N-methylformamido]-2-(pyridin-3-yl)acetic acid
4-[3-(pyrrolidine-1-sulfonyl)thiophene-2-carbonyl]-2-(trifluoromethyl)morpholine
4-(benzyloxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}butanamide
N-cyclopropyl-1-[1-(2,5-difluorobenzoyl)piperidin-4-yl]piperidine-4-carboxamide
1-(4-{5-methyl-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carbonyl}piperazin-1-yl)ethan-1-one
2-(4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,3,7-trimethyl-1H-indole
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)oxolane-3-carboxamide
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(pyridin-3-yloxy)propyl]acetamide
2-(4-{2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
5-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(2-fluorobenzoyl)-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-{4-[(2,5-dimethoxyphenyl)methyl]piperazine-1-carbonyl}-1-ethylpyrrolidin-2-one
4-chloro-2-[(1E)-3-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-methylprop-1-en-1-yl]phenol
2-[(3,4-dimethoxypyridin-2-yl)methyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one