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4-{[4-(carbamoylmethoxy)-3-chlorophenyl]methyl}-N,N-dimethylpiperazine-1-carboxamide
3-[1-methyl-5-(1-methylpiperidin-2-yl)-1H-1,2,4-triazol-3-yl]-1H-indole
2-{4-[4-(2-methylpropyl)piperazin-1-yl]quinazolin-2-yl}ethan-1-amine
4-({methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]amino}methyl)benzonitrile
4-fluoro-N-(2-{pyrazolo[1,5-a]pyrimidin-2-ylformamido}ethyl)benzamide
2-(1H-1,3-benzodiazol-1-yl)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-[1,3-dimethyl-4-(2-methylpiperidin-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-6-yl]pyridine
N-methyl-2-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
1-[(4-methoxyphenyl)methyl]-1-(oxolan-2-ylmethyl)-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
3-[(3S,4R)-1-(2-methylpropyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2,2-dimethylpropan-1-one
2-(4-methoxyphenyl)-N-(4-{4-[(3-methylbutyl)amino]piperidin-1-yl}phenyl)acetamide
5-{[2-(2-phenylethyl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
4-[4-(3,4-dimethylphenyl)-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
{3-[4-(1H-indol-2-ylmethyl)piperazin-1-yl]propyl}dimethylamine
5-ethyl-N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1,3,4-oxadiazol-2-amine
4-(1-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}piperidine-4-carbonyl)morpholine
2-[1-(3-methylphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(pyrimidin-4-ylmethyl)acetamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-2-(dimethylamino)-6-(4-methylthiophen-2-yl)pyridine-3-carboxamide
4-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-(6-methoxynaphthalen-2-yl)morpholine
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-cyclopropylethan-1-one
2-ethyl-8-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
2-{4-cyclohexyl-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
(2R,3R,6R)-5-(3-ethyl-1H-pyrazole-4-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(5-methanesulfonamido-2-methylphenyl)-3-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
1-{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
1-{4-[4-({[1-(morpholin-4-yl)cyclohexyl]methyl}amino)piperidin-1-yl]benzoyl}piperidin-3-ol
6-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-9H-purin-2-amine
2-{2-[4-(1-propyl-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,3-benzodiazole
5-(morpholin-4-ylmethyl)-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]furan-3-carboxamide
3-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]urea
3-[(dimethylamino)methyl]-1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}piperidin-3-ol
4-(4-{[(6,6-dimethyl-1-phenyl-4,5,6,7-tetrahydro-1H-indazol-4-yl)amino]methyl}phenyl)but-3-yn-1-ol
N-[1-({[(1-ethyl-1H-pyrazol-4-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]-2-(phenylsulfanyl)acetamide
N-cyclopentyl-5-methyl-N-[(4-methylphenyl)methyl]-1-propyl-1H-pyrazole-4-carboxamide
3-[({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1λ6-thiolane-1,1-dione
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-phenylbenzamide
1-(2-{[(2,3-difluoro-4-methylphenyl)methyl]amino}pyrimidin-4-yl)piperidin-3-ol
1-ethyl-5-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}piperidin-2-one
2-(1,4-diazepane-1-carbonyl)-6-(4-fluorophenyl)-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1λ6-thiomorpholine-1,1-dione
3-cyclopropaneamido-4-methyl-N-[(5-methylpyrazin-2-yl)methyl]benzamide
5-fluoro-2-[1-(1H-imidazol-4-ylmethyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
6-{[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}-2-methylpyrimidin-4-ol
5-(2-phenylethyl)-5-(1-{2-[3-(trifluoromethyl)phenyl]acetyl}piperidin-4-yl)imidazolidine-2,4-dione
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-N-(3-methoxypropyl)-5-methylthiophene-2-carboxamide
1-[(2-fluorophenyl)methyl]-N-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-amine
1-ethyl-4-[5-(3-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-3-methylpiperazin-2-one
N-(4-chloro-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}phenyl)acetamide