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2-[1-(2-phenylethyl)-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl]ethan-1-ol
N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]-2-[3-(thiophen-3-yl)-1H-pyrazol-1-yl]acetamide
4-[1-butyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-2,6-dimethylpyrimidine
3-[1-(adamantan-1-yl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methyloxane-2-carboxamide
N-({7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-fluorobenzamide
2-(2-amino-4-methyl-1,3-thiazol-5-yl)-N-{[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]methyl}acetamide
N-cyclohexyl-3-({[2-(methylsulfamoyl)phenyl]carbamoyl}amino)propanamide
[1-(2-methoxybenzenesulfonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
(3R,4R)-4-{methyl[2-(pyridin-2-yl)ethyl]amino}-1-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperidin-3-ol
1-(2-chlorophenyl)-4-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]piperazin-2-one
7-ethyl-2-[3-(4-methoxyphenyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
2-{[4-(1,3-dimethyl-1H-pyrazol-5-yl)-5-(2-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
5-{5-[1-(1H-pyrazol-1-yl)propyl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
(2S,4R)-1-[(3-chlorophenyl)methyl]-N,N-diethyl-4-{[(2-hydroxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
1-[5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N-(3-ethylphenyl)-4-(2-methoxyethyl)piperazine-1-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N'-(2-{1-[(3-methylthiophen-2-yl)methyl]piperidin-3-yl}ethyl)ethanediamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[(5-propylfuran-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
8-(pyridin-2-yl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-1-[4-(5-methylfuran-2-yl)benzoyl]-4-propylpyrrolidin-3-yl]acetamide
6-chloro-2-{2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
2-(2-hydroxyethyl)-9-(2-methyl-1,3-thiazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
(butan-2-yl)[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](pyridin-3-ylmethyl)amine
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[4-(2-fluorophenoxy)phenyl]-1-[(3-methoxyphenyl)methyl]piperidine-4-carboxamide
N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]cyclobutanecarboxamide
3-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1-[3-(sulfamoylmethyl)phenyl]urea
N,1-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
(1S,6R)-9-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-{5-[8-(trifluoromethyl)quinolin-4-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
1-[3-(2-methoxybenzoyl)piperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[2-(pyridin-3-yloxy)ethyl]piperidine-3-carboxamide
3-[3-(1H-imidazol-1-yl)propyl]-1-[2-methyl-3-(pyrrolidin-1-yl)phenyl]urea
5-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-cyclohexyl-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-pyrazole-4-carboxamide
(3S)-4-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-3-ethylmorpholine
(4aS,8aR)-6-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-[2-(pyridin-2-yl)ethyl]piperazine
4-{4-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
3-[5-(2H-1,3-benzodioxol-4-yl)-4-phenyl-1H-imidazol-1-yl]propan-1-ol
2-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N-ethylacetamide
4-(1-benzylpiperidine-2-carbonyl)-1-phenylpiperazin-2-one
1-{2-[(3R,5R)-3-(hydroxymethyl)-5-(morpholin-4-ylmethyl)piperidin-1-yl]-2-oxoethyl}piperidin-2-one
N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[2-(cyclohexylmethyl)morpholin-4-yl]-3-(pyridin-4-yl)propan-1-one
6-(aminomethyl)-2-(thiophen-3-yl)-3,4-dihydropyrimidin-4-one
2-(3,4-dimethoxyphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)acetic acid
1-(2-{[(2,3-difluoro-6-methoxyphenyl)methyl](methyl)amino}ethyl)cyclopentan-1-ol