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methyl (2S,4S,5R)-5-(4-chlorophenyl)-4-(cyclopentylcarbamoyl)-1,2-dimethylpyrrolidine-2-carboxylate
6-fluoro-2-{[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]methyl}quinolin-4-ol
3-(3-fluorophenyl)-5-(3-fluoropropyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
6-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
1-{2-[(3,4-difluorophenyl)methyl]-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}propane-1,2-dione
8-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]-2,8-diazaspiro[4.5]decan-3-one
2-(adamantan-1-yl)-N-methyl-N-(1H-pyrazol-5-ylmethyl)acetamide
1-[1-(2,6-difluoro-3-methoxybenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol
2,6-dimethoxy-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
4-cyano-N-[3-(3-methoxyphenyl)phenyl]piperidine-1-carboxamide
(1S,9S)-11-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
4-cyclobutanecarbonyl-9-methoxy-7-[5-(trifluoromethyl)pyridin-2-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(2,5-dimethylphenyl)methyl]-4-(2-methoxyethyl)-1,4-diazepan-5-one
ethyl 2-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-2-yl}acetate
1-benzyl-4-cyclobutanecarbonyl-1,4-diazepan-6-ol
5-[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-2-methyl-1,4-dihydropyridin-4-one
1-(propan-2-yl)-4-(pyridine-4-carbonyl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,1-dimethyl-1H-pyrrole-2-carboxamide
2-fluoro-N-(1-{[(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)carbamoyl]methyl}-1H-pyrazol-4-yl)benzamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(3-methoxypropanoyl)piperidine-4-carboxamide
1-(cyclopropylmethyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
1-{2-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]ethyl}pyrrolidin-2-one
2-(dimethylamino)-4-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrimidine-5-carboxamide
(butan-2-yl)[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl](pyridin-4-ylmethyl)amine
3-[4-(hydroxymethyl)phenyl]-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
3,4,4-trimethyl-1-(2-phenoxybenzoyl)pyrrolidin-3-ol
1-{4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-methoxypropan-1-one
{[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}({[3-(trifluoromethyl)phenyl]methyl})amine
1-(1H-imidazol-2-ylmethyl)-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
2-[3-cyclopropyl-5-(1H-1,2,3-triazol-5-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
N-(adamantan-1-ylmethyl)-1-ethyl-N-methyl-3-(4-methylpiperazine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(1H-1,3-benzodiazol-2-yl)-2-methoxy-6-(prop-2-en-1-yl)phenol
1-ethyl-N-[2-(4-fluorophenyl)ethyl]-N-[(3-methoxyphenyl)methyl]-1H-pyrazole-3-carboxamide
methyl 1-benzyl-3-cyclopropaneamido-5-{[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1S,5R)-3-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-[1-(3-methylbutyl)piperidin-4-yl]ethyl]methylamine
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methyl-4-oxo-3,4-dihydrophthalazine-1-carboxamide
5,6-dimethyl-2-[4-({methyl[(6-methylpyridin-2-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
{1-[(2-methyl-1H-imidazol-4-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-{[(1S)-1-phenylethyl]amino}piperidin-1-yl)benzamide
3-[(4aR,7aS)-6,6-dioxo-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
6-oxo-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}-1,6-dihydropyridine-2-carboxamide
4-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane-1-carbaldehyde
(3S,9aR)-8-(4-chlorobenzoyl)-3-(1H-imidazol-4-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-{[2-(3,4-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}-3-(2-methylpropyl)-1,2,4-oxadiazole
({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)(methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
(2S,4R)-4-amino-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidine-2-carboxamide
1-(5-chloropyridin-2-yl)-4-(2,3-dihydro-1H-indene-5-carbonyl)piperazine
N-(1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-2-methyl-1-oxopropan-2-yl)thiophene-2-carboxamide