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(4aS,8aR)-1-(3-hydroxypropyl)-6-(2-methoxypyridine-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
(3S,4S)-1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-4-propylpyrrolidine-3-carboxylic acid
N-[2-(1H-pyrrol-1-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
(1S,5R)-6-(2-methoxyethyl)-3-[2-(phenylsulfanyl)ethyl]-3,6-diazabicyclo[3.2.2]nonane
(4aS,7aR)-1-(3-hydroxypyridine-2-carbonyl)-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}pyrrolidin-2-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]acetamide
6-fluoro-N-methyl-N-(pyridin-2-ylmethyl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
{1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-ethylpiperidin-3-yl}methanol
2-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-6-methoxy-1-methyl-1H-indole
N-methyl-5-{[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]methyl}furan-2-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[3-(5-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperazine
2-{2-[2-(6-methyl-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
5-cyano-6-methyl-N-(3-methyl-1,2,4-thiadiazol-5-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-methyl-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
1-benzyl-4-[(4-fluoro-3-methylphenyl)methyl]-1,4-diazepan-6-ol
N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
2-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propane-1,3-diol
N-(2-methyl-1,3-benzothiazol-5-yl)-6-(3-oxo-2,3-dihydro-1H-indene-1-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
2-(pyridin-4-ylmethyl)-9-(pyrrolidine-1-sulfonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(3-methyl-4,5-dihydro-1,2-oxazol-5-yl)-1-phenyl-3-(2-phenylethyl)-1H-1,2,4-triazole
2-methyl-6-[1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-4-yl]-3,4-dihydropyrimidin-4-one
1-(4-benzylpiperazin-1-yl)-3-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl}propan-1-one
N-methyl-2-[methyl(2-phenylethyl)amino]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-[(3-ethoxy-3-oxopropyl)carbamoyl]piperidine-3-carboxylate
1-(2-{[(4-methylphenyl)methyl]carbamoyl}ethyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-{4-[(2-fluorophenyl)methyl]-1,4-diazepan-1-yl}propan-1-one
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1'-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-3-(3-fluorophenyl)benzamide
3-{[1-(oxolane-3-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-{[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methyl-4-[4-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)phenyl]but-3-yn-2-ol
1-(3-propylmorpholin-4-yl)-2-(quinazolin-4-yloxy)ethan-1-one
2-{[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]amino}-N-(pyrazin-2-yl)acetamide
1-(2-{1-[(5-methylthiophen-2-yl)sulfonyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
8-methoxy-2-[3-(3-methoxypropyl)piperidin-1-yl]quinoline
N4,N4,N6-trimethyl-N6-(quinolin-2-ylmethyl)pyrimidine-4,6-diamine
[1-(4-fluorophenyl)propyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-cyclopropylpyrazolo[1,5-a]pyrimidine-3-carboxamide
4-{[2-(1H-indol-3-yl)ethyl]amino}-N-(2-methoxyethyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
3-(1-{[5-(4-chlorophenyl)furan-2-yl]methyl}piperidin-3-yl)-1-(morpholin-4-yl)propan-1-one
2-amino-5-methyl-4-(2-methyl-1H-imidazol-4-yl)-6-(4-methylphenyl)pyridine-3-carbonitrile
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2-(naphthalen-2-yloxy)propanamide
(2R,3R)-3-(morpholin-4-yl)-1'-(1H-pyrrole-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-3-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}urea
2-(dimethylamino)-N-(1-{7-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
4-chloro-N-ethyl-2-fluoro-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)benzamide
7-cyclopentyl-2-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}-2,7-diazaspiro[4.5]decan-6-one
2-methoxy-N,4-dimethyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,3-thiazole-5-carboxamide