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1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-{[2-(5-methylfuran-2-yl)phenyl]methyl}piperazine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[3-(1H-imidazol-1-yl)propyl]acetamide
1-methyl-3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]urea
2-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
9-(cyclopropylmethyl)-1-methyl-4-[(1-propyl-1H-imidazol-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
5-methyl-N-[(1-methylpyrrolidin-3-yl)methyl]hexanamide
2-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
N-[2-(morpholin-4-yl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]cyclopropane-1-carbonitrile
N-[3-(1H-imidazol-1-yl)propyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
N-[(3R,4S)-1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]-2-hydroxyacetamide
N-[2-(2-fluorophenyl)ethyl]-5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
4-fluoro-N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)benzamide
2-[1-benzyl-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-2-yl]ethan-1-ol
N,6-dimethyl-N-[1-(pyridin-3-yl)propyl]imidazo[1,2-a]pyridine-2-carboxamide
1-[2-(dimethylamino)ethyl]-3-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-(3-methoxyphenyl)pyrrolidine-2,5-dione
8-fluoro-2-({[1-(pyridin-3-yl)propyl]amino}methyl)quinolin-4-ol
1-(1H-indazol-7-yl)-3-pentylurea
3-(4-chlorophenyl)-5-(2,3-dihydro-1,4-benzodioxine-2-carbonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyridine-3-carboxamide
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
methyl 2-[({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)carbamoyl]benzoate
3-(1,3-benzothiazol-6-yl)-1-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]urea
[1-(2-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}ethyl)piperidin-2-yl]methanol
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methyl-N-(propan-2-yl)piperidine-3-carboxamide
5-ethyl-2-methyl-4-[3-(1H-pyrazol-1-yl)phenyl]pyrimidine
N-(2-hydroxyethyl)-3-[(3S,4R)-1-(2-methylpropyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanamide
4-ethyl-3-[1-(2-phenoxybutanoyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-cyclohexyl-6-hydroxy-4-[3-(5-methylfuran-2-yl)butyl]-1,4-diazepan-2-one
1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)-2-(1H-1,2,3,4-tetrazol-5-yl)ethan-1-one
5-methoxy-3-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)-1H-indazole
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methanol
(4aS,8aR)-6-(4-amino-5-methylpyrimidin-2-yl)-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(4-fluoro-3-methylphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-ethyl-3-methyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-pyrazole-5-sulfonamide
N-[3-(2,3-dimethylphenoxy)propyl]-N-methyl-2-(1H-1,2,4-triazol-3-ylsulfanyl)acetamide
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(3,5-dimethoxyphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
(2S,4R)-4-amino-1-[2-(2-oxoazepan-1-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]-1-methyl-1H-pyrrole-3-carbonitrile
5-(azocane-1-carbonyl)-1-(2-methoxyethyl)-4-oxo-N-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-methyl-N-(pyridin-4-ylmethyl)piperidin-4-amine
N-(2,2-diphenylethyl)-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
9-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carbonyl}pyridine-2-carbonitrile
3-[methyl({2-[4-(3-methylpyridin-2-yl)piperazin-1-yl]pyrimidin-4-yl})amino]propane-1,2-diol
N-[2-(4-{[2-(4-chloro-2-methylphenoxy)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]oxolane-2-carboxamide
3-[1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
(3aS,6aS)-2-[(4,6-dimethylpyrimidin-2-yl)methyl]-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid