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1-[4-(3-fluorophenyl)phenyl]-N-(1H-1,2,4-triazol-5-ylmethyl)piperidin-4-amine
2-butyl-4-methyl-3-oxo-N-[3-(1,3-thiazol-4-yl)phenyl]piperazine-1-carboxamide
ethyl 1-{1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperidine-4-carboxylate
6-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-3-carboxamide
1-ethyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(2-methyl-1H-imidazol-1-yl)propanamide
7-[(3-hydroxy-6-methylpyridin-2-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-{2-oxo-8-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetic acid
2-amino-2,3-dimethyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)butanamide
(4aS,8aR)-6-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
N-[2-(dimethylamino)-1-phenylethyl]-N-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
1-[5-(dimethyl-1,3-thiazole-5-carbonyl)-1-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-(pyridin-4-ylmethyl)piperazine
5-methyl-3-(piperidin-4-yl)-3,4-dihydroquinazolin-4-one
4-({[2-(2-aminoethyl)-5,6-dimethylthieno[2,3-d]pyrimidin-4-yl]amino}methyl)-1-(2-methoxyethyl)pyrrolidin-2-one
1-[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-{4-[2-(4-chlorophenoxy)ethyl]phenyl}-5-methyl-1,3,4-oxadiazole
2-amino-3-ethyl-N-[1-(pyrazin-2-yl)piperidin-4-yl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-{3-[2-(2-methylphenyl)pyrrolidin-1-yl]propanamido}benzamide
1-(furan-2-ylmethyl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}piperidine-3-carboxamide
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-methyl-N-(propan-2-yl)acetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-amino-4-ethyl-1,3-thiazole-5-carboxamide
N-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
[1-(4-tert-butylbenzoyl)-3-[(2-fluorophenyl)methyl]piperidin-3-yl]methanol
4-(4-benzyl-1H-pyrazol-5-yl)-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
{7-fluoro-5-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
(1R,3s,6r,8S)-4-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
2-[1-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]pyridine
(3R,4S)-1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-amine
methyl({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
5-ethyl-5-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
N-(oxan-4-ylmethyl)-1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carboxamide
1-ethyl-2-oxo-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1,2-dihydropyridine-4-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-ethyl-N-propyl-1,2-oxazole-3-carboxamide
methyl 3-ethyl-2-(1H-pyrazol-3-yl)-3H-imidazo[4,5-b]pyridine-6-carboxylate
1-{2-[4-(4-hydroxyquinolin-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
3-[2-(methylsulfanyl)benzoyl]-1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidine
5-{2-[(1R,5S,8S)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 3-(2-chlorobenzenesulfonamido)-5-{[2-(3-methyl-1H-pyrazol-1-yl)acetamido]methyl}benzoate
1-[(2-chlorophenyl)methyl]-1-(2-hydroxyethyl)-3-(3-methyl-1-propyl-1H-pyrazol-5-yl)urea
(7-methoxy-3,7-dimethyloctyl)({2-[4-(propan-2-yl)piperazin-1-yl]ethyl})amine
2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoxaline
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-4-methoxybenzamide
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
7-(cyclopropylmethyl)-2-[2-(pyridin-2-ylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
7-[2-(1H-imidazol-2-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
9-(6-cyclopropylpyrimidin-4-yl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
ethyl 1-(ethanesulfonyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidin-4-ol
2-phenyl-5-[2-(trifluoromethyl)morpholine-4-carbonyl]-2,3-dihydro-1H-pyrazol-3-one
methyl({[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl})(pyrimidin-4-ylmethyl)amine