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4-[1-(furan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]-2-(propan-2-yl)pyrimidine
1-[(2-fluorophenyl)methyl]-N-(1H-indol-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(6-phenoxypyridin-3-yl)-1-(pyrazine-2-carbonyl)piperidine-4-carboxamide
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]piperidine-3-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-oxo-1-phenylpyrrolidine-3-carboxamide
8-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[2-(azocan-1-yl)-2-oxoethyl]-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidine-2,5-dione
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-7-fluoro-2-methylquinoline
2-(1,3-benzothiazol-2-ylmethyl)-4-[4-(4-propylpiperazine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-1-{3-[(2-methylprop-2-en-1-yl)oxy]phenyl}urea
3-({3-[3-(furan-3-yl)phenyl]-1H-pyrazol-1-yl}methyl)pyridine
2-[3-(furan-2-yl)-5-{3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propyl}-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-[(2-methoxyphenyl)methyl]-N-methyl-6-oxo-N-(2-phenoxyethyl)piperidine-3-carboxamide
5-(1,5-dimethyl-1H-pyrazol-4-yl)-1-(4-methoxyphenyl)-3-methyl-1H-1,2,4-triazole
3-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]propanamide
2-{4-[(2,4-difluorophenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-({3-[2-(3-fluorophenyl)ethyl]piperidin-1-yl}methyl)-5-methoxypyridin-4-ol
1-benzyl-8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl({[1-(2-methylpropyl)pyrrolidin-3-yl]methyl})(1,3-thiazol-2-ylmethyl)amine
2-({6-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidin-4-yl}amino)ethan-1-ol
(4aS,8aR)-1-propyl-6-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
methyl 1-[1-(4,6,7-trimethylquinazolin-2-yl)piperidin-4-yl]piperidine-2-carboxylate
N-[2-(dimethylamino)ethyl]-N-ethyl-1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
7-[(4-fluorophenyl)methyl]-2-(3-methylthiophene-2-carbonyl)-2,7-diazaspiro[4.5]decane
(4aR,8aR)-2-cyclopentanecarbonyl-7-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
2-(2-{[(2-phenyl-1,3-oxazol-4-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-cyclobutyl-4-[(1-phenylethyl)sulfamoyl]benzamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]acetamide
1-[(4-methoxyphenyl)methyl]-4-[2-(1H-1,2,4-triazol-5-yl)benzoyl]piperazin-2-one
2-(1,2-benzoxazol-3-yl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]acetamide
4-methyl-N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H-imidazole-5-carboxamide
N-(2-methoxyethyl)-N-(1,3-thiazol-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
5-[4-(2-hydroxyethyl)piperidine-1-carbonyl]-1-[2-(4-methoxyphenyl)ethyl]piperidin-2-one
{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
2-{5-[(2S)-1-methanesulfonylpyrrolidin-2-yl]-3-methyl-1H-1,2,4-triazol-1-yl}benzoic acid
1-(4-{4-[6-(4-methylthiophen-2-yl)-3-(piperidine-1-carbonyl)pyridin-2-yl]piperazin-1-yl}phenyl)ethan-1-one
N-(5-chloro-2-methoxyphenyl)-3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]propanamide
4-(2-methylpiperidine-1-carbonyl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine
2-(3-fluoro-4-hydroxyphenyl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
3-{1-[2-(2H-1,2,3-benzotriazol-2-yl)acetyl]piperidin-3-yl}-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-3-(4-methylphenyl)propan-1-one
1-(benzyloxy)-8-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
3-(2-amino-1,3-thiazol-4-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
5-(4-phenylpiperidin-1-yl)-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
3-[(3R,4S)-1-(1H-imidazol-4-ylmethyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
4-(5-{6-chloroimidazo[1,2-a]pyridin-2-yl}-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl)-1-methylpiperidine
N-{[3-methyl-7-(thiophene-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}pyrazine-2-carboxamide
1-(2-hydroxyethyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
ethyl 1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate