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3-methyl-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1-propyl-1H-pyrazole-4-carboxamide
4-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)benzoic acid
2-(2,3-dihydro-1-benzofuran-5-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
N-(adamantan-1-yl)-8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
3-methyl-N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
3-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1-(4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)urea
1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
4-{1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidine-3-carbonyl}morpholine
3-(3-fluorophenyl)-1-methyl-3-{2-oxo-2-[4-(quinazolin-4-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
1-(1-methyl-1H-pyrrol-2-yl)-2-{6-oxo-7-propyl-2,7-diazaspiro[4.5]decan-2-yl}ethane-1,2-dione
3-{4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
(3aS,6aS)-2-acetyl-5-(5-ethyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[2-(1-{5-cyclopropyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidin-4-yl)ethyl]dimethylamine
3-(benzyloxy)-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
4-(4-{[2-(1H-indol-1-yl)ethyl](methyl)amino}piperidin-1-yl)-N,6-dimethylpyrimidin-2-amine
2-(2-{[4-(2-amino-6-oxo-1,6-dihydropyrimidin-4-yl)piperazin-1-yl]methyl}phenoxy)propanoic acid
methyl 2-(benzylsulfamoyl)-6-[(2-methylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[1-hydroxy-2-({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)ethyl]phenol
2-(2-methoxyphenoxy)-N-[(1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)methyl]acetamide
5-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
4-(4-methyl-1H-pyrazol-1-yl)-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid
1-({2-methoxy-5-[3-(trifluoromethyl)phenoxy]phenyl}methyl)pyrrolidine
[1-(5-chloro-3-fluoropyridin-2-yl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
N-[2-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethyl]pyridine-3-carboxamide
2,5-dimethyl-3-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1-phenyl-1H-pyrrole
5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-3-(5-methylfuran-2-yl)-1H-pyrazole
(2S,4R)-N-cycloheptyl-1-[(3,4-difluorophenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
propyl (3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carboxylate
2-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
(3ar,6ar)-N-{[1-methyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-2-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
ethyl 1-(pyridin-3-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
3-(3-tert-butyl-1-phenyl-1H-pyrazol-5-yl)-1-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)urea
1-{1-[2-(dimethylamino)ethyl]-3-methyl-1H-pyrazol-5-yl}-3-[1-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]urea
N-ethyl-N-methyl-6-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-3-carboxamide
5-ethyl-5-[1-(3-hydroxybutyl)piperidin-4-yl]-3-[2-(4-methoxyphenyl)ethyl]imidazolidine-2,4-dione
4-[3-(3-methoxypyrrolidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]quinoline-6-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(4-ethylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylamino)acetamide
3-(1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-5-(propan-2-yl)-1,2-oxazole
1-ethyl-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-{[5-(4-ethoxyphenyl)furan-2-yl]methyl}-4-(4H-1,2,4-triazol-3-yl)piperidine
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-(diphenylmethyl)-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](pyridin-4-ylmethyl)amine
(1R,5R)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-{1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl}benzoic acid
5-(3,3-diphenylpiperidin-1-yl)-5-oxopentanamide