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5-[2-(dimethylamino)phenyl]pyridine-3-carboxamide
8-(5-ethoxy-2-methyl-1-benzofuran-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-{1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
(3R,9aR)-8-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-3-(propan-2-yl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(5-ethyl-1,2-oxazole-3-carbonyl)-4-(pyrrolidine-1-carbonyl)piperidine
1-[3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-[4-(furan-3-carbonyl)-1,4-diazepane-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
3-chloro-2-[3-(2-methoxyphenoxy)azetidin-1-yl]pyridine
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
(3aR,6aR)-2-[5-fluoro-4-(methylamino)pyrimidin-2-yl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(8-methyl-2-{4-[(2-methylphenyl)methyl]piperazin-1-yl}quinolin-3-yl)methanol
N-cyclopentyl-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
1-[(2E)-3-phenylprop-2-en-1-yl]-N-[3-(propan-2-yloxy)propyl]-1H-1,2,3-triazole-4-carboxamide
4-(1-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carbonyl)morpholine
1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3-(2-methylphenyl)pyrrolidin-3-ol
4-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridine
N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)propanamide
1-(4-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine-7-carbonyl}piperidin-1-yl)-2-ethoxyethan-1-one
N-{3-[4-({[3-(dimethylamino)phenyl]formamido}methyl)-5-methyl-1,3-oxazol-2-yl]phenyl}-5-methylthiophene-2-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-diazepane
1-(dimethylamino)-2-(4-{[4-(2-hydroxyethoxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)propan-2-ol
2-[(4-chlorophenyl)methyl]-8-cyclopentyl-2,8-diazaspiro[4.5]decan-3-one
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-2-(2-oxocyclopentyl)acetamide
N-(2-fluoro-4-methylphenyl)-2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}acetamide
5-chloro-2-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrimidine
6-{[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]amino}-N,N-dimethylpyrazine-2-carboxamide
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methylpropanamide
5-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-(4-fluorophenoxymethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-[3-(propan-2-yloxy)propyl]-1,3-oxazole-4-carboxamide
5-({7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)-2-methoxyphenol
(1S,2S,9S)-6-oxo-N-(2,4,6-trimethylpyridin-3-yl)-7,11-diazatricyclo[7.3.1.02,7]tridecane-11-carboxamide
N-ethyl-N-[1-(4-methoxyphenyl)propyl]-1-methyl-1H-1,2,3-benzotriazole-5-carboxamide
N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)furan-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-propyl-1,3-thiazole-4-carboxamide
(3aS,6aS)-2-acetyl-5-(4-cyclobutyl-6-methylpyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[3-(2-chlorophenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]-N-[(4-ethylphenyl)methyl]-N-methylacetamide
1-cyclohexyl-3-(2-fluorophenyl)-3-[2-(3-methoxypiperidin-1-yl)-2-oxoethyl]pyrrolidine-2,5-dione
1-{[4-(1-benzofuran-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-4-ol
[1-(4-chlorophenyl)ethyl]({[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
N-butyl-2-{imidazo[1,2-a]pyridin-3-yl}-N-(thiophen-3-ylmethyl)acetamide
N-(4-methylphenyl)-N'-{[4-(pyrrolidin-1-ylmethyl)phenyl]methyl}propanediamide
6-methyl-1-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-(trifluoromethyl)-1,2-dihydropyridin-2-one
1-[1-(2-phenylethyl)-5-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-1,4-diazepan-5-one
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
5-[3-(3-fluorophenyl)-1H-pyrazol-4-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
(2S,4R)-4-amino-N-methyl-1-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]pyrrolidine-2-carboxamide
4-{6-[1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-3-yl]-2-methylpyrimidin-4-yl}morpholine
5-(azepan-1-yl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide