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3-[4-(4-acetylphenyl)piperazine-1-carbonyl]piperidine-1-carboxamide
methyl 1-[(3S,5S)-1-[(4-chlorophenyl)methyl]-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-methyl-2-(3-methyl-1,2-oxazol-5-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
1-cyclopentyl-N-methyl-N-[2-(4-methylphenoxy)ethyl]-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[2-(6-oxo-3-phenyl-1,4,5,6-tetrahydropyridazin-1-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
1-ethyl-3-[2-oxo-2-(piperidin-1-yl)ethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
3-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
4-[3-(3-chlorophenoxymethyl)-5-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
1-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
N-[(1S)-1-(3-methylpyridin-2-yl)ethyl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
2-amino-1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-methylpropan-1-one
3-(azocan-1-yl)-1-(4-benzyl-6-hydroxy-1,4-diazepan-1-yl)propan-1-one
1-cyclobutanecarbonyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}piperidine-4-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-1-(pyrimidin-2-yl)piperidin-4-amine
1-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]cyclopropane-1-carboxamide
N-[4-(4-{[2-(4-fluorophenyl)ethyl]amino}piperidin-1-yl)phenyl]cyclopentanecarboxamide
N-butyl-7-[(4-fluorophenyl)methyl]-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
ethyl 1-{5-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperidine-4-carboxylate
2-{3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}ethan-1-ol
3-[(4-fluorophenyl)methyl]-5-methyl-5-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
5-[1-(1H-indole-6-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-[(1-propyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-{[4-(methylsulfanyl)phenyl]methyl}-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
(1R,5S)-N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
1-(2-cyclopropylpyrimidine-5-carbonyl)-4-(2-hydroxyethyl)-1,4-diazepan-6-ol
ethyl 2-[4-(2-cyclopropyl-1,3-benzoxazole-6-carbonyl)morpholin-3-yl]acetate
N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-N5-tert-butyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
6-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-[(1E)-pent-1-en-1-yl]benzoic acid
1-(2-{4-[2-(methoxymethyl)pyrimidin-5-yl]-1H-1,2,3-triazol-1-yl}ethyl)pyrrolidin-2-one
1-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrrolidin-2-one
9-[(1-propyl-1H-imidazol-2-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methoxyethyl)-1-{1-[2-(4-methylphenoxy)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
ethyl 4-(2-oxo-1-phenylpyrrolidine-3-amido)piperidine-1-carboxylate
3-(2H-1,3-benzodioxole-5-carbonyl)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
4-[(2-chloro-4-fluorophenyl)methyl]-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-(1-methoxybutan-2-yl)piperidine-3-carboxamide
(1R,6S)-3-(4-chloro-2-methylbenzoyl)-9-methyl-3,9-diazabicyclo[4.2.1]nonane
5-(3-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(1H-pyrazol-1-yl)butanamide
4-{4-[3-(1-methoxyethyl)phenyl]-1H-pyrazol-5-yl}pyridine
4-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methoxypyridine-3-carbonitrile
1-(3-chlorothiophene-2-carbonyl)-4-[(3-fluorophenyl)methyl]-1,4-diazepan-5-one
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carboxamide
1-(2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetyl)-1,4-diazepan-5-one
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(4-fluorophenyl)-1-{1-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}ethyl]methylamine
N,N-dimethyl-1-(pyridine-2-carbonyl)azepan-4-amine
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
8-(3-ethoxypropanoyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one