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2-amino-3-ethyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
3,3-dimethyl-4-(morpholin-4-ylmethyl)-1-(thiophene-2-sulfonyl)piperidin-4-ol
3-[(dimethylamino)methyl]-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)pyrrolidin-3-ol
5-cyclopropanecarbonyl-1'-(2-methyl-1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-(propan-2-yl)acetamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
2-methoxy-5-{[methyl({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)amino]methyl}phenol
(1R,3S)-7-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
3-(1H-pyrazol-1-yl)-N-{3-[(pyridin-3-yl)amino]propyl}benzamide
8-[2-(2,5-dimethoxyphenyl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
3-(3-fluorophenyl)-6-(2-methoxybenzoyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-cyclopropyl-3-({2-[(trifluoromethyl)sulfanyl]ethyl}sulfamoyl)benzamide
5-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}pyridine-2-carbonitrile
1-(cyclopropylmethyl)-N-ethyl-5-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-[(4-fluorophenyl)methyl]-5-[1-(6-hydroxypyridine-3-carbonyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)imidazolidine-2,4-dione
6-({4-phenyl-5-[1-(pyridin-2-yl)-1H-pyrrol-2-yl]-1H-imidazol-1-yl}methyl)pyrimidin-4-ol
6-(6-hydroxy-4-{[5-(hydroxymethyl)furan-2-yl]methyl}-1,4-diazepan-1-yl)pyrazine-2-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-3-carboxamide
3-(3-chlorothiophene-2-carbonyl)-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
(2R,6R)-4-[2-(2-hydroxyethoxy)ethyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-(1-{[2-(cyclopentyloxy)phenyl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
2-[1-(propane-1-sulfonyl)pyrrolidin-2-yl]-1,3-benzothiazole
4-[4-(diethylamino)benzoyl]-1-(2-methylphenyl)piperazin-2-one
(1R,9S)-5-amino-3-[2-(propylsulfanyl)pyrimidin-5-yl]-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
2-(furan-2-yl)-N-(thiolan-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(2,3-dihydro-1H-isoindol-2-yl)-N-[2-(piperidin-1-yl)ethyl]pyridine-2-carboxamide
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-1-ethylpiperidine-3-carboxamide
2-(2-hydroxypropanoyl)-N-(2-phenoxyethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-(1-{7-[(2,3-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
methyl 1-[(3S,5S)-1-[(4-acetamidophenyl)methyl]-5-{[3-(methylsulfanyl)phenyl]carbamoyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
6-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-1-benzoxepine-4-carboxamide
1-(2-fluorophenyl)-2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethan-1-ol
2-{[(2-methoxyphenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-(diethylamino)-1-[3-(2-methoxybenzoyl)piperidin-1-yl]ethan-1-one
N-[5-(4-benzylpiperidine-1-carbonyl)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl]furan-2-carboxamide
2-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pyridine-4-carboxamide
3-({4-[3-(2-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)pyridine
N-methyl-4-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-4'-ylmethyl}benzamide
(1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-ethylpiperidin-3-yl)methanol
N-(2-{[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}ethyl)acetamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[4-(pyridin-2-yl)butyl]acetamide
4-(4-{[2-(morpholin-4-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl)benzamide
4-amino-5-(8-hydroxyquinolin-2-yl)-2-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-7-one
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-2-(pyridin-4-yl)pyridine
3-{5-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
2-ethyl-8-(2-{methyl[(4-methylphenyl)methyl]amino}acetyl)-2,8-diazaspiro[4.5]decan-3-one
ethyl 6-[2-methyl-4-(2-methylpropyl)-3-oxopiperazin-1-yl]pyridine-3-carboxylate
4-(4-{1-[(3,4-dimethylphenyl)methyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
1-[(2-chloro-6-fluorophenyl)methyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane