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1-{2-[2-(2,3,4-trimethoxyphenyl)-1H-imidazol-1-yl]ethyl}piperidine
N-(1-{7-[2-(2-chlorophenyl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-3-methoxypropanamide
3-(1H-indol-3-yl)-1-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propan-1-one
2-(2,3-dimethylphenoxy)-1-{4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}ethan-1-one
2-chloro-6-fluoro-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
methyl N-[1-({[5-(dimethylcarbamoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}carbamoyl)ethyl]carbamate
3-cyclohexyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
3-[(2-chlorophenyl)methyl]-N-[1-(4-methoxyphenyl)ethyl]-N-methyl-1,2-oxazole-5-carboxamide
N-[(3S,4R)-4-propyl-1-{[2-(trifluoromethoxy)phenyl]methyl}pyrrolidin-3-yl]acetamide
2-({2-[butyl(4-hydroxybutyl)carbamoyl]phenyl}amino)acetic acid
3-[4-(2-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
2-{2-[(4-fluorophenyl)methyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-6-methylpyridine
3-{[(1-cyclohexylpiperidin-4-yl)methyl]carbamoyl}-5-methoxybenzoic acid
5-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-1,3-benzothiazole
5-{4-[(8-methoxy-2H-chromen-3-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
2-(cyclopropylmethyl)-7-[2-(1-ethylpiperidin-4-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-cyclopropyl-5-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
1-{4-[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]piperidin-1-yl}ethan-1-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-(oxan-4-yl)piperidine-3-carboxamide
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-3-(morpholine-4-sulfonyl)benzamide
2-{1-[2-(2-chloro-4-fluorophenyl)ethyl]piperidin-2-yl}ethan-1-ol
1-(2-chloroprop-2-en-1-yl)-7-(methylsulfanyl)-3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,2-dihydroquinolin-2-one
N-({1-[(2,5-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-3-methylfuran-2-carboxamide
1-{2-[(2,1,3-benzoxadiazol-4-ylmethyl)(methyl)amino]ethyl}piperidin-2-one
(1R,3S)-3-(2-aminoethoxy)-7-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-3-[(2-fluoroethyl)sulfamoyl]benzamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[2-(1H-imidazol-2-yl)benzoyl]piperidine
2-methoxy-5-(pyridin-4-yl)benzamide
N-[2-(4-ethylphenoxy)ethyl]-N-methyl-2-(1,2,3,6-tetrahydropyridin-4-yl)acetamide
6-fluoro-2-{9-oxa-2-azaspiro[5.5]undecan-2-ylmethyl}quinolin-4-ol
2-(phenylamino)-N-{2-[(pyridin-3-yl)amino]ethyl}pyrimidine-5-carboxamide
4-(2-butyl-1H-imidazol-4-yl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
3-{1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}-N-[(3,4-difluorophenyl)methyl]propanamide
2-(2,4-dimethoxyphenyl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethan-1-one
1-acetyl-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(3S,4S)-1-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
3-fluoro-2-methoxy-N-methyl-N-(oxan-2-ylmethyl)benzamide
[3-propyl-1-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperidin-3-yl]methanol
(4aS,8aR)-6-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
(2R,3R,6R)-5-(isoquinoline-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(5-amino-1H-1,2,4-triazol-3-yl)-1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]propan-1-one
N-butyl-3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-methylbenzamide
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[3-(pyridin-3-yloxy)propyl]acetamide
N-[1-(7-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-3-methylbutyl]-2-methoxyacetamide
5,7-dimethyl-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}pyrido[2,3-d]pyrimidin-4-amine
methyl 9-(cyclopentyloxy)-7-oxo-3-(pyridin-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-ethyl-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]pyrimidine-5-carboxamide
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)[1-(pyridin-3-yl)ethyl]amine