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ethyl 4-[3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanoyl]piperazine-1-carboxylate
1-methyl-3-phenyl-8-[2-(pyrrolidin-1-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
2-({6-[3-(3-methoxybenzoyl)piperidin-1-yl]pyrimidin-4-yl}amino)ethan-1-ol
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)cyclopent-3-ene-1-carboxamide
1-[(2-methoxyphenyl)methyl]-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}piperidin-2-one
(2R)-2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidine
3-phenyl-N-[1-(7-{[4-(propan-2-yloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]propanamide
N-methyl-2-(methylsulfanyl)-N-[1-(2-phenylethyl)piperidin-3-yl]benzamide
(1S,6R)-3-[(4-methanesulfonylphenyl)methyl]-3,9-diazabicyclo[4.2.1]nonane
N-butyl-2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(propan-2-yl)acetamide
5-{2,7-dimethylpyrazolo[1,5-a]pyrimidin-5-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
6-(4-chlorophenyl)-N-(1-methoxybutan-2-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
7-methoxy-3-{[4-(6-methylpyridin-2-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-(4-{[2-(1H-imidazol-2-yl)ethyl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}(pyridin-4-ylmethyl)amine
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-4-yl}methyl)-2-(3-fluorophenyl)-N-methylacetamide
7-(1,3-benzothiazol-2-yl)-4-[(3,4-difluorophenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
7-(cyclopropylmethyl)-2-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-2,7-diazaspiro[4.5]decan-6-one
1-(5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)piperidine
N-methyl-2-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,2-dihydroquinoline-4-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]oxane-4-carboxamide
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-N-methylpropanamide
2-[4-(6,7-dimethoxy-4-methylquinolin-2-yl)piperazin-1-yl]ethan-1-ol
2-({[(3R,4R)-4-(hydroxymethyl)-1-[(4-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
7-(5-chloropyridin-2-yl)-4-(4-fluorobenzenesulfonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(1-{[1-(propane-2-sulfonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(1H-imidazol-1-yl)ethan-1-one
(2R)-2-amino-1-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pentan-1-one
1-cyclohexyl-4-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}piperazin-2-one
ethyl 1-[2-(2-chlorophenyl)ethyl]-1H-imidazole-2-carboxylate
2-methyl-4-(4-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenyl)butan-2-ol
ethyl 3-[(2-fluorophenyl)methyl]-1-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]piperidine-3-carboxylate
4-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-[(2S,4R)-2-(diethylcarbamoyl)-4-(2-methyl-1H-pyrrole-3-amido)pyrrolidin-1-yl]acetic acid
1-(3-phenylpropyl)-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]piperidin-2-one
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-4-(2,4-dioxoimidazolidin-1-yl)benzamide
1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
N-[3-methoxy-4-(3-methylbutanamido)phenyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
2-(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
ethyl 2-({[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)amino)acetate
3-chloro-N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}pyridine-4-carboxamide
N-[3-(benzyloxy)phenyl]-9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
(5S,9aS,9bS)-2-(3-methoxyphenyl)-5-(2-phenylethynyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-[2-(ethylsulfanyl)ethyl]-4-(1H-imidazol-1-yl)benzamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
4-(1-benzyl-3-phenyl-1H-1,2,4-triazol-5-yl)-1λ6-thiane-1,1-dione
N-[1-(4-{4-[hydroxy(thiophen-2-yl)methyl]piperidine-1-carbonyl}phenyl)-1H-pyrazol-4-yl]oxane-4-carboxamide
N-(furan-2-ylmethyl)-N-(2-hydroxyethyl)-1-methylazepane-2-carboxamide
3-methoxy-5-[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]benzoic acid
(1S,5R)-3-[(dimethylcarbamoyl)methyl]-N-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide