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3-[(3S,4R)-1-(2-methylpropyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-1-(piperidin-1-yl)propan-1-one
(2E)-4-methyl-1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}pent-2-en-1-one
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyridin-3-ylmethyl)piperazine
8-(2,4-dimethylpyrimidine-5-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
7-(1-benzothiophen-3-yl)-4-(4-methyl-1,3-oxazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[2-(5-methylfuran-2-yl)ethyl]-4-(pyridin-3-yl)pyrimidin-2-amine
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-(4-chloro-2-methylbenzoyl)-1-[3-(1H-imidazol-2-yl)benzoyl]piperidine
5-(2,6-difluorophenoxymethyl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
4-{[5-(3,6-dimethylpyrazin-2-yl)-2-hydroxyphenyl]methyl}piperazine-1-carbaldehyde
1-[cyclohexyl(methyl)amino]-3-(2-{[(2-methoxyethyl)amino]methyl}phenoxy)propan-2-ol
[4-benzyl-1-(pyridin-3-ylmethyl)piperidin-4-yl]methanol
3-{[(2,3-dihydroxypropyl)(methyl)amino]methyl}-6-ethoxy-1,2-dihydroquinolin-2-one
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-hydroxy-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
4-{3-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-2,2-dimethylpropyl}morpholine
5-(4-chloro-2-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
6-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
4-[(2-methoxyethyl)amino]-N,5-dimethyl-N-[1-(1,3-thiazol-2-yl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
2-[3-(2-methoxybenzoyl)piperidin-1-yl]pyridine-4-carbonitrile
(4aS,7aR)-1-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-methyl-1-(2-methylphenyl)-4-[3-(pyrazin-2-yl)propanoyl]piperazin-2-one
4-methyl-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
N-[4-chloro-3-({[2-(2-oxopyrrolidin-1-yl)ethyl]carbamoyl}amino)phenyl]-2-methoxyacetamide
(3S,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(3-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(cyclopropylmethyl)-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-chloro-4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methylquinoline
(2S,4R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
N-methyl-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-N-(2-phenylethyl)piperidin-3-amine
[(3R,4R)-4-[(dimethylamino)methyl]-1-(2,2-diphenylethyl)pyrrolidin-3-yl]methanol
6-(2-fluorophenyl)-2-(3-{[methyl(oxan-4-yl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(2R,4S)-1-[(8-chloroquinolin-2-yl)methyl]-4-hydroxypiperidine-2-carboxylic acid
3-(4-methoxyphenyl)-3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propan-1-ol
(4aS,7aR)-1-{2-[4-(dimethylamino)phenyl]acetyl}-4-ethyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{1-[2-(3-chlorophenyl)acetyl]piperidin-3-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
1-{2-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}piperidin-2-one
N-[(2-methoxyphenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 8-(naphthalen-2-ylmethyl)-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
ethyl 1-({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)piperidine-4-carboxylate
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N,N-diethylacetamide
N-{1-[1-(6-methylquinoline-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
2-({[(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amino}methyl)-3-methoxyphenol
3-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-{[1-(5-chloropyridin-2-yl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
[4-(oxan-2-ylmethyl)-1-(thiophene-3-sulfonyl)piperidin-4-yl]methanol
1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
3-{2-[(5-{3-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}pyridin-2-yl)amino]ethyl}-1,3-oxazolidin-2-one
methyl 3-acetamido-5-{[(4-ethoxyphenyl)methyl]amino}-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
6-[3-(acetamidomethyl)piperidin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
5-{1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}isoquinoline