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3-(morpholin-2-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
2-methyl-5-(3-methylphenyl)-4-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-3-yl}pyrimidine
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(furan-2-yl)ethyl]benzamide
3-[2-(dimethylsulfamoyl)ethyl]-1-(2,3,4-trifluorophenyl)urea
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methylpyridin-2-yl)methyl]acetamide
methyl 1-(2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}acetyl)piperidine-4-carboxylate
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl){[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}amine
1-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-3-[3-ethyl-4-(4-fluorophenyl)-1-methyl-1H-pyrazol-5-yl]urea
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]acetamide
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-1-phenylcyclohexane-1-carboxamide
5-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
1-[1-(cyclopentylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
3-[(4-fluorophenyl)methyl]-5-[1-(1H-indole-5-carbonyl)piperidin-4-yl]-5-methylimidazolidine-2,4-dione
1-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
1-{2-[({2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}amino)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-4,4-dimethylpiperidine-1-sulfonamide
{1-[(3-methyl-1H-pyrazol-5-yl)methyl]-4-(3-phenylpropyl)piperidin-4-yl}methanol
N-[(2-fluorophenyl)methyl]-3-[1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl]propanamide
{[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl}bis(prop-2-en-1-yl)amine
N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
(1S,4S)-3,3-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-methylidenebicyclo[2.2.1]heptane-1-carboxamide
1-[(4-fluorophenyl)methyl]-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)propanamide
[(5-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-4-ethyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
4-(1H-pyrazol-4-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]butanamide
N-[2-(4-cyclohexylmorpholin-2-yl)ethyl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-(3,5-dimethyl-1H-pyrazol-4-yl)-1,2,4-oxadiazole
N-[(2S,4R,6R)-2-(6-chloro-2-fluoro-3-methylphenyl)-6-(propan-2-yl)oxan-4-yl]acetamide
methyl 3-(2,4-difluorobenzoyl)-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-{9-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-N-(2-phenylethyl)piperidin-3-amine
N-(2-hydroxyethyl)-1-{1-[1-(trifluoromethyl)cyclopropanecarbonyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-[(naphthalen-1-ylmethyl)amino]-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
(3S,7S)-5-(3-fluoropyridin-4-yl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]-6-(1-methyl-1H-imidazol-2-yl)pyridazine
(4-{[({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)(methyl)amino]methyl}oxan-4-yl)methanol
1-tert-butyl-N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-5-oxopyrrolidine-3-carboxamide
{7-[6-(morpholine-4-carbonyl)pyrazin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
1-({4-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]phenyl}methyl)-1H-1,2,3,4-tetrazole
4-(hydroxymethyl)-1-[(3-methylthiophen-2-yl)methyl]azepan-4-ol
4-ethyl-3-(piperidin-4-yl)-1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(5-{[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,4-triazol-3-yl)pyridine
2-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]pyridin-3-ol
7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decane
2-(4-chlorophenyl)-N-(6-chloropyridin-3-yl)morpholine-4-carboxamide
methyl({[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl})({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
2-[(1H-imidazol-2-ylmethyl)(methyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-({4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}methyl)pyridine-3-carboxylic acid