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N-[(5-methylpyrazin-2-yl)methyl]-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
1-(2-phenoxyethyl)-4-[3-(thiophen-2-yl)-1H-pyrazole-4-carbonyl]piperazine
N-{3-[1-(3-chloro-2-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]propyl}acetamide
(1s,4s)-N-({1-[(3-fluoro-2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-4-hydroxycyclohexane-1-carboxamide
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(2-ethoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(3-phenoxyazetidin-1-yl)sulfonyl]-N-(propan-2-yl)benzamide
N-[(3S,4R)-1-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]-4-propylpyrrolidin-3-yl]acetamide
methyl 2-(2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-methylacetamido)acetate
2-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-N-[2-(2-methoxyphenyl)ethyl]acetamide
1-({5-[1-(cyclohexylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)-4-methylpiperazine
N-cyclopentyl-4-[5-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-3-(1H-pyrazol-1-yl)benzamide
N-tert-butyl-3-{[4-(propan-2-yl)phenyl]amino}piperidine-1-carboxamide
2-cyclopropyl-1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
1-{4-[hydroxy(pyridin-2-yl)methyl]piperidin-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-{[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-4-methoxyphenol
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]acetamide
1-(2-methoxy-5-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
N-(1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxybenzamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](propyl)(pyridin-3-ylmethyl)amine
5-[(2E)-but-2-en-2-yl]-4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazole
5-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
(2S,4S)-N-ethyl-1-(naphthalen-1-ylmethyl)-4-[(pentan-3-yl)amino]pyrrolidine-2-carboxamide
2-(1-benzofuran-5-yl)-1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazole
6-chloro-N-({1-[ethyl(methyl)amino]cyclopentyl}methyl)-1-methyl-1H-indole-2-carboxamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({[(5-methyl-1,2-oxazol-3-yl)methyl]amino}methyl)piperidin-2-one
ethyl (2S)-2-(2-{[(2-chlorophenyl)methyl]sulfanyl}acetamido)propanoate
4-[(4-methoxy-3-methylphenyl)methyl]-3-(2-oxo-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethyl)piperazin-2-one
2-(dimethylamino)-1-[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(3-methylphenyl)ethan-1-one
2-methyl-N-{1-[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
3-(2-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}-2-oxoethyl)-2-sulfanylidene-1,3-thiazolidin-4-one
{5-fluoro-7-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
2-methyl-3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-4,5,6,7-tetrahydro-1H-indol-4-one
(1R,5R)-3-(2,3-dimethyl-1H-indole-7-carbonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-[1-(4-chlorophenyl)cyclobutyl]-1-(2-methoxyacetyl)piperidine-3-carboxamide
1-[1-(cyclohexylmethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
2-(propan-2-yl)-9-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-N-[(1-ethylpyrrolidin-3-yl)methyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
{[3-chloro-5-methoxy-4-(prop-2-en-1-yloxy)phenyl]methyl}[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]amine
2-benzyl-9-(6-hydroxyhexyl)-2,9-diazaspiro[5.5]undecan-3-one
4-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperazin-2-one
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
N-[2-(7-{[5-(methoxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-4-methylbenzamide
3-[(dimethylamino)methyl]-1-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}piperidin-3-ol
1-[4-(3-{[(4,6-dimethoxypyrimidin-2-yl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2,3-difluoro-N-(oxolan-2-ylmethyl)benzamide
1-cyclopropanecarbonyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidine-4-carboxamide