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1-(2-cyclohexylethyl)-3-hydroxy-3-({[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]amino}methyl)piperidin-2-one
3-(2-amino-1,3-thiazol-4-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-methyl-N-{1-[1-(4-methyl-2-oxopentanoyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-2-(1H-pyrazol-1-yl)acetamide
N-{2-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-2-oxoethyl}benzamide
(3S,4S)-1-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
1-(1-benzothiophen-2-ylmethyl)-3-(1,3,4-thiadiazol-2-yl)urea
N-(3-benzamido-4-methoxyphenyl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
2-methyl-5-(3-{[(6-phenylpyridazin-3-yl)amino]methyl}pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-{[6-(3-chlorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-(2-methoxyethyl)oxolane-2-carboxamide
5-(3-cyclohexyl-1H-pyrazol-4-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-(3-{[(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}-1H-indol-1-yl)acetamide
1-(4,6-dimethylquinazolin-2-yl)-N-[2-(2-fluorophenyl)ethyl]piperidin-4-amine
{[3,5-dichloro-4-(prop-2-en-1-yloxy)phenyl]methyl}[1-(pyrazin-2-yl)propan-2-yl]amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(3-methyl-1,2-oxazol-5-yl)acetamide
3-(2,5-dihydro-1H-pyrrol-1-ylmethyl)-N-(2-methyl-1H-1,3-benzodiazol-6-yl)benzamide
N-{[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]methyl}-4-fluoroaniline
1-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
(1s,4s)-4-{[methyl({[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}cyclohexan-1-amine
N-(2-{7-[(2-phenyl-1,3-thiazol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
2-[2-(butan-2-yl)phenoxy]-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}acetamide
7-methoxy-3-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1H-3-benzazepine
(4aS,8aR)-1-(3-aminopropyl)-6-{pyrazolo[1,5-a]pyridine-3-carbonyl}-decahydro-1,6-naphthyridin-2-one
1-(3-phenylphenyl)-N-[2-(1,3-thiazol-4-yl)ethyl]piperidin-4-amine
6-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyridine-2-carbonitrile
4-{4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
(2R)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
2-[2-chloro-5-(trifluoromethyl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
N-{1-[1-(cyclobutylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
1-[(5-ethylfuran-2-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
4-(3-chloro-2-methylbenzenesulfonyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
{2-oxo-2-[2-(2-phenylethyl)piperidin-1-yl]ethyl}urea
1'-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]spiro[indene-1,4'-piperidine]
[1-(2,3-dihydro-1H-inden-2-yl)-3-[(3-methoxyphenyl)methyl]piperidin-3-yl]methanol
methyl 4-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidine-1-carbonyl}benzoate
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(morpholin-4-yl)ethan-1-one
2-amino-4-(dimethyl-1,2-oxazol-4-yl)-5-methyl-6-phenylpyridine-3-carbonitrile
1-methyl-8-{[4-(methylsulfanyl)phenyl]methyl}-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2-methoxy-5-{4-[1-(morpholin-4-yl)ethyl]phenyl}phenyl)methanol
4-(5-chloropyridine-2-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(pyridin-2-ylmethyl)piperazine
1-{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-ol
(4aR,8aS)-1-(3-ethoxypropyl)-6-[(4-methoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
1-({4-methyl-5-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}-N-[1-(pyrimidin-4-yl)ethyl]benzamide
1-(4-{[3-(4-cyclopentylpiperazine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}-3-methoxyphenyl)ethan-1-one
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-1-(4-chlorophenyl)methanesulfonamide
1-{2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propyl}-3,5-dimethyl-1H-pyrazole
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}propanamide
[(4-ethylphenyl)methyl](methyl){[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
4-fluoro-N-(2-{[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)benzamide