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3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3,4-dihydro-2H-1-benzopyran-6-carbonyl)piperidine
1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
4-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-3-fluorobenzonitrile
N-[1-(1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
2-cyclopropyl-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1,3-benzoxazole-6-carboxamide
1-(3-methyl-1H-pyrazole-5-carbonyl)-4-[(3-methylphenyl)methyl]piperazine
2-{[(3S,5S)-5-[4-(adamantan-2-yl)piperazine-1-carbonyl]-1-[(3-chlorophenyl)methyl]pyrrolidin-3-yl]sulfanyl}-4-methylpyrimidine
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(methylsulfanyl)benzamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-[(1-benzylpiperidin-4-yl)methyl]-2-cyclopropyl-N,4-dimethylpyrimidine-5-carboxamide
2-[2-(dimethylamino)ethyl]-9-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
methyl 2-[(cyclohexylmethyl)sulfamoyl]-6-[2-(methylsulfanyl)acetyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-methyl-N-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}oxolan-3-amine
3-[1-(morpholin-4-ylmethyl)cyclopentyl]-1-[4-(1H-pyrazol-1-yl)phenyl]urea
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl})methylamine
1,3-dimethyl-N-{[8-(2-methylpropyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-1H-pyrazole-5-carboxamide
N-[1-(3-fluorophenyl)-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-2-(methylamino)acetamide
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
2-[3-(2-chlorophenyl)-1-methyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-(propan-2-yl)acetamide
(3S)-1,3-dimethyl-4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
2-[5-(2,3-dimethoxyphenyl)-4-phenyl-1H-imidazol-1-yl]-3-methylbutan-1-ol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-methyl-N-[1-(pyridin-3-yl)pentyl]acetamide
1-{3-[2-(azetidin-1-ylmethyl)-6-methoxyphenoxy]propyl}-1H-imidazole
1-(cyclohexylmethyl)-5-(2-{[(4-fluorophenyl)methyl]amino}ethyl)pyrrolidin-2-one
(1S,4S)-2-{3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzoyl}-2-azabicyclo[2.2.1]heptane
7-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-2-oxa-7-azaspiro[4.5]decan-8-one
7-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-2-oxa-7-azaspiro[4.5]decan-8-one
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)methylamine
5-(methoxymethyl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}thiophene-2-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-3-(1H-pyrazol-4-yl)benzamide
1-cyclohexanecarbonyl-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
1-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-4-phenylpyrrolidin-2-one
(2E)-N-{[5-(4-methanesulfonylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(thiophen-2-yl)prop-2-enamide
benzyl N-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
1-{2-[2-(2,3-dimethoxy-5-methylphenyl)phenoxy]ethyl}-1H-imidazole
N-[(3,5-dimethoxyphenyl)methyl]-1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidin-4-amine
2-(2,2-dimethylpropanoyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
6-{1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]piperidin-3-yl}-2-methylpyrimidin-4-ol
3-fluoro-2-methoxy-N-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
(2R,6S)-2,6-dimethyl-4-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}morpholine
N-[(1-methyl-2,3-dihydro-1H-indol-5-yl)methyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
(3S,4S)-1-[(6-ethoxypyridin-3-yl)methyl]-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
5-(2,4-difluorophenoxymethyl)-N-[2-(1H-indol-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-8-fluoro-4-oxo-1,4-dihydroquinoline-2-carboxamide
2-(2-chlorophenyl)-3-methyl-N-[2-(pyrrolidin-1-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
ethyl 4-{2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperazine-1-carboxylate
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-methylpiperazine-1-sulfonamide
ethyl 4-[1-(2-oxo-4-phenylbutanoyl)piperidin-3-yl]piperazine-1-carboxylate
methyl[1-(4-methylpyridin-2-yl)propan-2-yl](quinolin-2-ylmethyl)amine