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N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N,N-diethyl-1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
2-(2-{[3-(dimethylamino)piperidin-1-yl]methyl}-4-(pyrazin-2-yl)phenoxy)acetic acid
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(4-methanesulfonylphenyl)ethan-1-one
N-(furan-2-ylmethyl)-3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carboxamide
2-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)oxane-2-carboxamide
4-{[4-(2,2-dimethylpropyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}phenol
3-fluoro-N-{1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
2-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
(2S)-2-amino-N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-hydroxypropanamide
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-3-methoxy-2,2-dimethylpropanamide
1-(diphenylmethyl)-N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
1-{1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]piperidin-4-yl}-1,4-diazepan-5-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(3-methylpyridin-4-yl)methyl]pyridin-2-amine
2-methyl-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}pyrido[2,3-d]pyrimidin-4-amine
N-{2-[4-(propan-2-yl)morpholin-2-yl]ethyl}-1H-indazole-3-carboxamide
8-[2-(1H-indol-1-yl)acetyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-methylpiperidin-3-yl)methyl]-4-oxo-N-(2-phenylethyl)pentanamide
N4-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-5-methylpyrimidine-2,4-diamine
1-{2-[3-cyclopropyl-1-(2-methoxyphenyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydropyridin-2-one
N-(propan-2-yl)-1-[(1s,4s)-4-(2,5-dimethoxybenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-[2-(4-fluorophenyl)ethyl]-4-[(5-propylpyrimidin-4-yl)amino]pyrrolidin-2-one
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]methylamine
(5S,9aS,9bS)-2-cyclopentyl-5-[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-(1-{1-[4-(1H-1,2,4-triazol-1-yl)phenyl]ethyl}-1H-1,2,3-triazol-4-yl)pyrimidine
1-ethyl-3-(propan-2-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
3-{1-[(3-chlorophenyl)methyl]azetidin-3-yl}pyridine
3-[({1-[(5-methylfuran-2-yl)methyl]piperidin-3-yl}oxy)methyl]pyridine
N-(1-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
(3R,5S)-N3-(4-fluorophenyl)-1-(naphthalen-2-ylmethyl)-N5-(oxolan-2-ylmethyl)piperidine-3,5-dicarboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]propanamide
N-[(2-fluorophenyl)methyl]-2-{4-[3-(1H-pyrrol-1-yl)propanoyl]morpholin-3-yl}acetamide
(3S,4S)-4-cyclopropyl-1-[3-(pyridin-4-yl)propanoyl]pyrrolidine-3-carboxylic acid
4-(piperazine-1-sulfonyl)-N-(thiolan-3-yl)benzamide
1-(4-{4-methyl-5-[(4-methylpiperazin-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(1H-1,2,3-triazol-1-yl)ethan-1-one
1-cyclohexyl-N-methyl-4-oxo-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
1-[3-(2-methoxybenzoyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-2-(pyrrolidine-1-carbonyl)piperazine
13-(7-methoxy-2H-1,3-benzodioxol-5-yl)-4,6-dimethyl-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
1-{1'-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
2-{1-[(2-fluorophenyl)methyl]-4-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
(3S,4R)-1-[(5-methylfuran-2-yl)methyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
(isoquinolin-5-ylmethyl)(methyl){[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}amine
4-[4-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
7-chloro-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-3,4-dihydroquinazolin-4-one
N-cyclopropyl-1-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-1,2,3-triazole-4-carboxamide
1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-propoxyethan-1-one