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N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
(1S,4S)-5-[(2S)-3-hydroxy-2-(methylamino)propanoyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-(4-{2,8-diazaspiro[4.5]decan-2-ylmethyl}phenyl)acetamide
5-{[(5-methyl-1-propyl-1H-pyrazol-4-yl)formamido]methyl}thiophene-2-carboxylic acid
1-methyl-N-[3-methyl-1-(pyridin-3-yl)butyl]-3-propyl-1H-pyrazole-5-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
5-(morpholin-4-ylmethyl)-8-{[5-(trifluoromethyl)pyridin-2-yl]oxy}quinoline
1-{4-[2-(2-methoxyethyl)piperidin-1-yl]piperidin-1-yl}butan-1-one
(4aS,7aR)-1-(5-chloropyridine-3-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-6-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-yl)-3,4-dihydropyrimidin-4-one
1-(furan-3-ylmethyl)-4'-propyl-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-(cyclopropylmethyl)pyridin-2-amine
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]acetamide
2-(1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
3-{2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
{[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
ethyl 4-[(2-chlorophenyl)methyl]-1-cyclopentanecarbonylpiperidine-4-carboxylate
N-[(3-cyclohexyl-1,2,4-oxadiazol-5-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
9-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
3-methyl-5-[2-(2-methyl-1H-imidazol-1-yl)propyl]-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}propanamide
2-(3-chloro-4-hydroxyphenyl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]acetamide
5-[(diethylcarbamoyl)methyl]-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-ethyl-4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-methylpyrimidine
3-hydroxy-1-(3-phenylpropyl)-3-{[(piperidin-4-ylmethyl)amino]methyl}piperidin-2-one
N-ethyl-4-oxo-1-(2-phenylethyl)-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
(4aR,7aS)-1-propanoyl-4-(1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[4-(dimethylamino)benzoyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
3-[1-(2-hydroxyethyl)-3-(1H-indol-3-yl)-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroisoquinolin-1-one
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-{[4-(trifluoromethoxy)phenyl]methyl}propanamide
8-chloro-3-[2-(4-phenylpiperidin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
3-(tert-butylsulfamoyl)-5-(cyclohexylamino)-N-[(1-methylpiperidin-3-yl)methyl]benzamide
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]acetamide
{1-[2-chloro-5-(trifluoromethyl)benzoyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
N-[(2R,3R)-1'-[(2,6-dimethoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-7H-pyrrolo[2,3-d]pyrimidin-4-amine
(1S,4S)-5-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[1-(7-{[3-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-phenoxyacetamide
N-[(2R,3R)-1'-(3-ethynylbenzoyl)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
N-[(7-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]oxolane-3-carboxamide
1-(2-fluorophenyl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-4,6-dimethylpyrimidin-2-amine
5-ethoxy-N-[(2-methyl-1,3-thiazol-4-yl)methyl]furan-2-carboxamide
N-methyl-2-[4-(methylsulfanyl)phenyl]-N-(1H-pyrazol-3-ylmethyl)acetamide
N-(4-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide