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1-ethyl-8-[(1-methyl-1H-indol-3-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-propanoylphenoxy)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-({1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}methyl)benzoic acid
{3-[({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)methyl]-2,4,6-trimethylphenyl}methanol
N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-1,1-dioxo-3,4-dihydro-2H-1λ6,2-benzothiazine-3-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[(2-methoxyethoxy)methyl]-3-(propan-2-yl)-1H-1,2,4-triazole
methyl 9-[(1-methylpiperidin-3-yl)methoxy]-7-oxo-3-{[4-(propan-2-yloxy)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-cyclopropyl-5-(2,3-dimethoxyphenyl)-1-methyl-1H,4H-pyrazolo[3,4-d]imidazole
2-ethyl-N-[2-(4-fluorophenyl)ethyl]pyrimidine-5-carboxamide
N-butyl-N-[(2-fluorophenyl)methyl]-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
1-{3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}-4-(2-methoxybenzoyl)piperazine
2-[(6-methylpyridin-2-yl)methyl]-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
3,5-dimethyl-N-{2-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}benzamide
N,N,2-trimethyl-7-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
[(3aS,6aS)-2-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
2-(dimethylamino)-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-(2-fluorophenyl)acetamide
3-{[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
1-(furan-2-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-2-yl)piperidine-4-carboxamide
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(4-fluorophenoxy)ethan-1-one
1,3-dimethyl-N-({8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1H-pyrazole-5-carboxamide
3-(dimethylsulfamoyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]-5-[(propan-2-yl)amino]benzamide
N-cyclohexyl-2-[1-(2-methoxyethyl)-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)pyrimidin-4-yl]pyrrolidin-3-ol
2-[3-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
(1R,9aR)-1-{[(1-methanesulfonylpiperidin-4-yl)amino]methyl}-octahydro-1H-quinolizin-1-ol
N-ethyl-N-[2-(3-methylphenoxy)ethyl]-3-(2-oxoimidazolidin-1-yl)benzamide
(3R,4R)-1-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-ethylpiperidine-3,4-diol
methyl 2-(4-{[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]carbamoyl}-2-oxopiperazin-1-yl)acetate
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-methyl-4-(quinoxaline-2-carbonyl)piperazin-2-one
(2S,4R)-1-benzyl-N-ethyl-4-[2-(2-methylphenyl)acetamido]pyrrolidine-2-carboxamide
1-(2-methoxybenzoyl)-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylic acid
methyl (2S,3S)-2-[(1-{4-[(dimethylsulfamoyl)amino]phenyl}piperidin-4-yl)amino]-3-methylpentanoate
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
2-(2-phenylethyl)-9-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
4-[4-(4-fluorophenyl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-1,2-dihydroquinolin-2-one
1-{6-hydroxy-4-[4-(methylamino)pyrimidin-2-yl]-1,4-diazepan-1-yl}-2-phenylethan-1-one
2-methoxy-N-(1-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
[(4-chloro-1-methyl-1H-pyrazol-3-yl)methyl](2-methoxyethyl)[(3-methylthiophen-2-yl)methyl]amine
N-{1-[(3-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-fluoropyridine-4-carboxamide
(4aR,7aS)-1-benzyl-4-(oxane-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(4-acetylpiperazin-1-yl)-6-methylquinolin-3-yl]methyl}-N-[2-(cyclohex-1-en-1-yl)ethyl]-2,5-dimethoxybenzamide
(1R,3S)-3-{[(4-hydroxyphenyl)methyl](pyridin-4-ylmethyl)carbamoyl}cyclopentane-1-carboxylic acid
3-[4-(2-methoxybenzoyl)piperazine-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-2H-indazole
2-methoxy-3-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}pyrazine
1-(6-methylpyridin-2-yl)-4-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperazine
N-[(8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]acetamide
(4aS,8aR)-6-(4-aminopyrimidin-2-yl)-1-(2-ethoxyethyl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
1-(2-ethoxyphenyl)-4-{1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperazine
3-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1-(pyrrolidin-1-yl)propan-1-one