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2-amino-6-(4-hydroxy-2-methylphenyl)-4-[1-(propan-2-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-3-[2-(2-methylphenyl)ethyl]piperidine
(2R)-2-{[5-(2-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}-4-methylpentanamide
N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]-2-(pyridin-3-yl)acetamide
N-(isoquinolin-5-ylmethyl)-2-methoxy-N,4-dimethyl-1,3-thiazole-5-carboxamide
5-{4-oxo-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl}pyridine-2-carbonitrile
1-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-(quinolin-5-yl)pyridine-3-carboxamide
N-ethyl-N-(1-hydroxypropan-2-yl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-[(2S)-2-hydroxy-3-phenylpropanoyl]-1-(2-methylphenyl)piperazin-2-one
(1S,5R)-3-[2-(2-chloro-4-fluorophenyl)acetyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-4-oxobutane-1-sulfonamide
(3aS,6aS)-2-cyclopentanecarbonyl-5-[(4-methyl-1,3-thiazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)sulfamoyl]diethylamine
{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}(methyl)(1,3-thiazol-2-ylmethyl)amine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-methylpropanamide
N'-({1-[(3,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)ethanediamide
2-[methyl(1,2-oxazol-3-ylmethyl)amino]-2-[3-(trifluoromethoxy)phenyl]acetic acid
3-[(3,4-difluorophenyl)methyl]-9-methoxy-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
N4-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-N2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-[2-(2,6-dichlorophenyl)ethyl]-4-hydroxy-1-methylpiperidine-4-carboxamide
1-phenoxy-2-[4-(pyridin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
2-amino-4-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-methoxy-6-({3-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)phenol
(1R,2R)-1-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-2,3-dihydro-1H-inden-2-ol
1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-4-yl)piperazine
3-({[4-(pyridin-3-yl)pyrimidin-2-yl]amino}methyl)-1,2,4-oxadiazole-5-carboxamide
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(pyridin-4-yl)propan-1-one
2-[5-(1-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)-1H-pyrazol-3-yl]acetic acid
1-{3-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
4-[3,5-dimethyl-1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
1-{1-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}-4-phenylpiperazine
1-ethyl-N-[(4-phenyloxan-4-yl)methyl]-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyridin-4-yl)piperazine
5-(1-cyclopentylpyrrolidin-2-yl)-N-methyl-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]thiophene-2-carboxamide
1-(2-methylpropyl)-N-(pyridin-4-ylmethyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-tert-butyl-1-methyl-4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
2-({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(2-hydroxyethyl)amino)ethan-1-ol
1-(1,4-dioxan-2-ylmethyl)-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
6-{[benzyl(ethyl)amino]methyl}-N-[(2-chlorophenyl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
(3aS,6aS)-2-(2,5-dimethylfuran-3-carbonyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
1-(3-{3-[(4-benzylpiperidin-1-yl)methyl]phenoxymethyl}piperidin-1-yl)-2-(1H-pyrazol-1-yl)ethan-1-one
{3-[(3-chlorophenyl)methyl]-1-(3-methylbenzenesulfonyl)piperidin-3-yl}methanol
2-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}-1-(pyridin-3-yl)ethan-1-ol
N,N,2-trimethyl-4-{[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
N-[3-(pyridin-4-yl)propyl]-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-[(4-fluorophenyl)methyl]pyrrolidine-2-carboxylate