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2-{[6-({[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}amino)pyrimidin-4-yl]amino}ethan-1-ol
2-(2H-1,3-benzodioxol-5-yl)-5-fluoro-1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
2-(5-tert-butyl-2H-1,2,3,4-tetrazol-2-yl)-N-(1-cyclopentyl-3-methyl-1H-pyrazol-5-yl)acetamide
4-methoxy-1-{[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}piperidine
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3S)-4-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-1,3-dimethylpiperazin-2-one
2-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-5-sulfamoylbenzamide
ethyl[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
5-(2-oxo-2-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-methyl-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-N-(1H-pyrazol-5-ylmethyl)-1,3-oxazole-4-carboxamide
8-(1-methyl-1H-pyrazole-4-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(4-{[2-(furan-2-yl)phenyl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecan-11-yl)propan-1-one
3-[(3R,4S)-1-(7-fluoro-4-methylquinolin-2-yl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
4-[3-(3-methoxyphenoxy)azetidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-{1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
ethyl 4-({[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}amino)piperidine-1-carboxylate
9-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-4-methyl-1-oxa-4,9-diazaspiro[5.5]undecan-3-one
N-[(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)methyl]-3-hydroxypyridine-2-carboxamide
1,5-dimethyl-4-({4-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-1-yl}methyl)-1H-pyrrole-2-carbonitrile
2-(2,5-dimethyl-1-phenyl-1H-pyrrole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxylic acid
1-[4-({2-[2-(dimethylamino)ethoxy]-3-methoxyphenyl}methyl)piperazin-1-yl]-2,2-dimethylpropan-1-one
7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3-(oxolan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(2,3-dihydro-1H-inden-2-yl)benzamide
2-{4-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]phenyl}-2-methylpropanamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-(furan-2-yl)-2-oxoacetamide
5-acetyl-N-[1-(3-phenylpropyl)piperidin-3-yl]thiophene-3-carboxamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(1-methyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-methyl-1-(3-oxo-3-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propyl)-1,2-dihydropyridin-2-one
2-{3-[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]phenoxy}acetamide
11-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-7-methyl-3,7,11-triazaspiro[5.6]dodecane
2-hydroxy-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-3-methylbutan-1-one
2-(3-fluoro-4-methoxyphenyl)-N,N-dimethylpyridine-3-carboxamide
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}[2-(3,4-dimethoxyphenyl)ethyl]methylamine
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-(2-phenylethyl)pyrrolidin-2-one
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-2-(2-methoxyethoxy)ethan-1-one
3-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-N,N-dimethylaniline
2-{4-[(5-ethylfuran-2-yl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
2-[3-(3,4-dimethoxyphenyl)-1H-indazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
(3S,4S)-4-(dimethylamino)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-ol
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-2,6-dimethylpyrimidine-4-carboxamide
N-(1-{1-[2-(2-methoxyphenyl)acetyl]piperidin-4-yl}-2-phenylethyl)-N-methyl-2-(1H-pyrazol-1-yl)acetamide
N-benzyl-N-(cyclopropylmethyl)-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[2-(3-fluorophenyl)ethyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
2-(3,5-difluorophenyl)-N-(oxolan-3-yl)acetamide
2-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-benzyl-5-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)-1H-1,2,3,4-tetrazole
1-[4-(4-{[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
N-cyclopropyl-2-[4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)piperidin-1-yl]acetamide