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1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-8-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-tert-butyl-1-(3-methylbutyl)-4-oxo-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
methyl 1-({4-[(2-chloro-3,4-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-2-carboxylate
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-ol
6-cyano-N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]pyridine-3-carboxamide
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pent-4-enamide
N-[2-(pyrazin-2-yl)ethyl]-6-[4-(trifluoromethyl)phenyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-(3-ethyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}urea
1-[(2-fluorophenyl)methyl]-4-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperazin-2-one
4-[(2-{1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]piperidin-3-yl}-1H-imidazol-1-yl)methyl]pyridine
5-[(3-fluorophenyl)methyl]-3-(2-hydroxyethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
(1S,3R)-N1-(1,3-benzoxazol-2-ylmethyl)-1,N2,N2,3,3-pentamethylcyclopentane-1,3-dicarboxamide
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3-fluorophenyl)methyl]-N-(2-methoxyethyl)pyrrolidine-2-carboxamide
(3S,4R)-1-[2-(1H-1,3-benzodiazol-1-yl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
{2-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]phenyl}methanol
2-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]benzonitrile
9-[(2,2-dimethyloxan-4-yl)methyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
dimethyl[(4-{1-[(6-methylpyridin-2-yl)methyl]piperidin-2-yl}phenyl)methyl]amine
1-ethyl-4-[({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]pyrrolidin-2-one
[(3R,5R)-1-(5-ethyl-1H-pyrrole-2-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-(1-tert-butyl-1H-pyrazol-4-yl)-N,3,6-trimethyl-N-(propan-2-yl)quinoline-4-carboxamide
N-(1,3-benzoxazol-2-ylmethyl)-N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}acetamide
5-(3-propyl-1,2,4-oxadiazol-5-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
3-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-2-methyl-1H-indole
({4-ethyl-5-[1-(5-fluoropyridine-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
7-methyl-6-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1H,2H-pyrazolo[1,5-a]pyrimidin-2-one
4-{5-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}phenol
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,5-dimethyl-1H-1,2,4-triazole
N-[(2-fluorophenyl)methyl]-1-methyl-5-[4-(morpholin-4-yl)piperidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-[3-(propan-2-yl)-1H-pyrazol-1-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N-methyl-N-(thiophen-3-ylmethyl)pyridin-2-amine
N-[(2-aminopyridin-3-yl)methyl]-2,5,6-trimethylpyrimidin-4-amine
N-[(1-{[1-(carbamoylmethyl)-1H-indol-3-yl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
2-(3-methoxyphenoxymethyl)-N-methyl-N-(pyridin-3-ylmethyl)-1,3-oxazole-4-carboxamide
methyl 4-[(4-{2-cyclohexyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)methyl]benzoate
N-[1-(cyclohexylmethyl)piperidin-3-yl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-[2-(dimethylamino)ethyl]-N-methyl-1-[4-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-3-amine
1-ethyl-N-methyl-6-oxo-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
3-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-methyl-5-(2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-(1H-imidazol-4-ylmethyl)pyrrolidine-3-carboxylic acid
6-ethyl-2-methyl-N-[1-(pyridin-3-yl)propan-2-yl]quinoline-4-carboxamide
{imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
4-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]benzene-1-sulfonamide
3-{1-[1-(2,5-dimethylfuran-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-methylphenyl)urea
[1-(1H-imidazol-1-yl)propan-2-yl]({[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl})amine
ethyl 1-[2-(phenoxymethyl)-1,3-oxazole-4-carbonyl]piperidine-4-carboxylate
8-fluoro-2-[(4-hydroxyazepan-1-yl)methyl]quinolin-4-ol
N,1-dimethyl-2-oxo-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,2-dihydroquinoline-4-carboxamide