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(2S,4R)-1-[(4-methoxy-3-methylphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-methyl-N-(1H-pyrazol-5-ylmethyl)pyrrolidine-2-carboxamide
3-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
2-amino-4-[2-(pyrrolidin-1-yl)pyrimidin-5-yl]-6-(thiophen-3-yl)pyridine-3-carbonitrile
N-(quinolin-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
methyl 3-[(4-methoxy-3-methylphenyl)methyl]-7-oxo-9-(pyridin-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}pentane-1,5-diamine
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N,7,8-trimethyl-N-(propan-2-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
N-{2,5-dimethyl-3-[4-phenyl-1-(thiophen-2-ylmethyl)-1H-imidazol-5-yl]-1H-pyrrol-1-yl}acetamide
1-(2-methoxyethyl)-3-(propan-2-yl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(5-amino-1H-pyrazole-3-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
[2-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)phenyl]methanol
3-benzoyl-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidine
1-[1-(3,4-dichlorophenyl)-1H-1,2,4-triazol-5-yl]-6-azaspiro[2.5]octane
7-(5-chloro-2-methoxyphenyl)-4-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(2,6-difluorophenyl)methyl]-N-methyl-N-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3-benzothiazole-2-carboxamide
(1R,7S)-N-ethyl-3-[(4-fluorophenyl)methyl]-4-oxo-N-(pyridin-4-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
ethyl 4-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-1H-pyrazole-4-carbonyl)piperazine-1-carboxylate
1-(4-fluorophenyl)-4-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
3-{1-[2-(naphthalen-2-yl)acetyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
6-(2-methylpropyl)-4-[3-(naphthalene-1-carbonyl)piperidine-1-carbonyl]-1,2-dihydropyrimidin-2-one
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)morpholine-4-sulfonamide
4-(4-cyclopentylpyrimidin-2-yl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-[1-(7-{[4-(2-methylpropyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]pyridine-3-carboxamide
methyl 8-[(2-methoxynaphthalen-1-yl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-[1-(pyridin-2-yl)propan-2-yl]-1H-1,3-benzodiazole-7-carboxamide
6-fluoro-2-{4-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]piperidin-1-yl}-4-methylquinazoline
1-(2-methoxyacetyl)-N-[(1-phenylcyclohexyl)methyl]piperidine-4-carboxamide
N-[(1S,2S)-1,3-dihydroxy-1-phenylpropan-2-yl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
1-phenyl-4-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]piperazin-2-one
N-{[7-chloro-2-(2,5-dimethoxyphenyl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]acetamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-{[3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}acetic acid
methyl[(4-methyl-1H-imidazol-2-yl)methyl][(2,4,6-trimethoxyphenyl)methyl]amine
N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)but-3-enamide
4-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-1-phenylpiperazin-2-one
5-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2-(pyridin-3-yl)pyrimidine
8-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
7-methyl-4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
1-[2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]piperidine-4-carboxamide
ethyl 2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}pyridine-3-carboxylate
8-methoxy-N-(4,4,4-trifluorobutyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(2-ethoxyphenyl)methyl]-3-hydroxy-N-(prop-2-en-1-yl)propanamide
methyl 1-{2-hydroxy-3-[4-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[3-(pyridin-2-yl)propyl]piperidine-3-carboxamide
3-[5-(4-methylphenoxymethyl)-1,3,4-thiadiazol-2-yl]-1-(oxan-3-ylmethyl)urea
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]acetamide
3-methyl-1-(2-{[(4-methylphenyl)methyl]sulfanyl}phenyl)-3-(1-methylpyrrolidin-3-yl)urea
methyl (2S)-3-carbamoyl-2-(2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamido)propanoate
N-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide