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6-{4-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
4-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3aR,7aS)-2-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-2,3,3a,4,7,7a-hexahydro-1H-isoindole
1-cyclopropanecarbonyl-N-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidin-3-amine
1-cyclohexyl-4-[(2-fluoro-5-methoxyphenyl)methyl]piperazin-2-one
[1-({1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanamine
5-chloro-2-(2-{[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1H-pyrrol-1-yl)pyridine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-5-(2-methoxyacetamido)-N-methyl-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-cyclopentylpropanamide
1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}-N,N-dimethylpyrrolidin-3-amine
(4aS,7aR)-1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(5-chlorothiophen-2-yl)methyl]-1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
methyl(quinolin-6-ylmethyl){[4-({1-[2-(trifluoromethyl)benzenesulfonyl]piperidin-4-yl}oxy)phenyl]methyl}amine
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-2-(4-methanesulfonylphenyl)acetamide
(2S)-4-({4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}formamido)-2-hydroxybutanoic acid
(1S,5R)-3-methyl-6-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(1H-indol-3-yl)acetamide
N-[2-(3-methoxyphenyl)-1-[1-(3-methylbutanoyl)piperidin-4-yl]ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
3-(furan-2-yl)-1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}propan-1-one
1-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
methyl 7-oxo-9-(pyridin-2-ylmethoxy)-3-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-{4-[4-({[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]benzoyl}piperidin-3-ol
N-(3-fluorophenyl)-1-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]benzoic acid
2-[methyl(pyridin-3-ylmethyl)amino]-1-{1-oxa-8-azaspiro[4.5]decan-8-yl}ethan-1-one
2-[3-(2-methylbutyl)-5-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-1-yl]acetic acid
5-[2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]pyridin-3-amine
4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}benzonitrile
N-[(3R,4S)-4-cyclopropyl-1-(3-fluoropyridin-2-yl)pyrrolidin-3-yl]propane-1-sulfonamide
N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-cyclopentyl-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
4-(4-methanesulfonylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
4-{[6-hydroxy-4-(1H-pyrazole-4-carbonyl)-1,4-diazepan-1-yl]methyl}benzamide
2-{[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](furan-2-ylmethyl)amino}butan-1-ol
N-methyl-1-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)piperidine-2-carboxamide
4-chloro-2-({1-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-6-azaspiro[2.5]octan-6-yl}methyl)phenol
4-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}pyridin-3-ol
1-[(4aR,8aS)-1-[4-(3-fluorophenyl)benzoyl]-decahydro-1,6-naphthyridin-6-yl]-3-(pyridin-3-yl)propan-1-one
[(2-chloro-4-fluorophenyl)methyl]({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-(2,5-difluorophenyl)-N-{[8-(furan-3-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(4-methyl-1,4-diazepan-1-yl)acetamide
3-(4-methoxy-3,5-dimethylbenzoyl)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine
4-(2,3-dihydro-1,4-benzodioxin-6-yl)furo[3,2-c]pyridine
2-{1-[(2-ethoxyphenyl)methyl]-4-(pyridine-4-carbonyl)piperazin-2-yl}ethan-1-ol
8-{1-[2-(dimethylamino)ethyl]-3-methyl-1H-pyrazole-5-carbonyl}-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
2-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-5-{[3-(4-methoxy-3,5-dimethylbenzoyl)piperidin-1-yl]methyl}phenol
4-(2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-4-carbonyl)morpholine
1-(2-{[1-(cyclohex-1-en-1-yl)ethyl]amino}-4-methylpyrimidin-5-yl)ethan-1-one