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4-({1-benzyl-5-[1-(2-methyl-1H-imidazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl}methyl)-1-methylpiperidine
N-[1-(4-fluorophenyl)ethyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
1-[(4-methyl-1H-imidazol-5-yl)methyl]-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
2-amino-6-(2-fluorophenyl)-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-2-(5-oxopyrrolidin-2-yl)acetamide
3-ethyl-N-{[7-(3-methoxybenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
1-methyl-6-oxo-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1,6-dihydropyridine-3-carboxamide
1-(benzenesulfonyl)-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
4-methyl-2-propyl-6-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]pyrimidine
1-[4-(2-methoxyethyl)piperazin-1-yl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}ethan-1-one
2-{5-[2-(benzylsulfanyl)ethyl]-3-ethyl-1H-1,2,4-triazol-1-yl}acetic acid
4-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-2-one
[3-(3-methoxypropyl)-1-[2-methyl-2-(morpholin-4-yl)propyl]piperidin-3-yl]methanol
N-[2-(3-chlorothiophene-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}-2-(morpholin-4-yl)acetamide
8-(6-aminopyridine-3-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
6,7-dimethyl-4-[({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}amino)methyl]-2H-chromen-2-one
methyl 7-oxo-3-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-9-(thiophen-2-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
5-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-[2-(3,4-difluorophenyl)ethyl]-1-(5-propyl-1,2-oxazole-4-carbonyl)piperidine
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
1-{1-[1-(9H-purin-6-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}cyclopentan-1-ol
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
4-(2,2-dimethylpropyl)-3-(2-oxo-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}ethyl)piperazin-2-one
N-(2H-1,3-benzodioxol-5-yl)-1-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
2-[2-(dimethylamino)ethyl]-9-(1-methyl-1H-pyrazole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(5-fluoro-2-methylbenzoyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
2-(4-fluorophenyl)-1-{[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
2-{methyl[2-(morpholin-4-yl)ethyl]amino}-2-[4-(methylsulfanyl)phenyl]acetic acid
5-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidine-1-carbonyl]-2-methylphenol
1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
methyl 3-[(3S,4R)-1-[(4-fluorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
1-(2-amino-6-methoxypyrimidin-4-yl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-methyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-{1-[(3-methoxyphenyl)methyl]-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
1-[(2-ethoxyphenyl)methyl]-3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]piperidine
N-(4-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}phenyl)acetamide
{1-[4-(4-{[(3,4-dimethoxyphenyl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-yl}methanol
1-{4-[(1,3-dihydroxy-2-methylpropan-2-yl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
1-(carbamoylmethyl)-N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]piperidine-4-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
N,N-dimethyl-2-{[5-(propan-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]formamido}propanamide
(4aS,8aR)-1-(2-aminoethyl)-6-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
5-(3-phenylpropyl)-5-{1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
1-cyclopentanecarbonyl-3-(3-methoxypropyl)piperidine-3-carboxylic acid
[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl](methyl){[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine