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2-benzyl-4-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-1,3-thiazole
5-(2H-1,3-benzodioxole-5-carbonyl)-3-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-methyl-N-[(4-methylphenyl)methyl]benzamide
9-methoxy-3-(naphthalen-2-ylmethyl)-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-(6-methylpyridine-3-carbonyl)-N-[4-(propan-2-yl)phenyl]piperidin-3-amine
4-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-1-(propan-2-yl)-1H-pyrazole
4-(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)pyrimidin-2-amine
N-[(2R,3R)-1'-cyclohexanecarbonyl-2-ethoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-(pyridin-4-yl)piperazine
2-[1-(2-methylpropyl)-4-(3-propyl-1H-pyrazole-5-carbonyl)piperazin-2-yl]ethan-1-ol
1-methyl-5-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}-1H-imidazole
2-(2H-1,3-benzodioxol-5-yl)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]ethan-1-one
1-(1-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}propyl)-1H-pyrazole
(3S,4S)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
N,N-diethyl-1-{6-[(2-methoxyethyl)amino]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}pyrrolidin-3-amine
2-methyl-1-{4-[(2E)-4-methylpent-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-1-ol
2-{4-[4-(dimethylamino)-5-methylpyrimidin-2-yl]phenoxy}acetic acid
7-(cyclopropylmethyl)-2-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decane
4-(1H-indol-5-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
1-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
N-{1-[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
7-[(3-methylphenyl)methyl]-2-[(3,4,5-trimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane
1-{4-[(3-aminoazepan-1-yl)methyl]thiophen-2-yl}ethan-1-one
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-{6-methyl-2H-[1,3]dioxolo[4,5-g]quinolin-8-yl}piperidine
1-(butan-2-yl)-N3-ethyl-4-oxo-N5-[(1-phenylcyclohexyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-(5-chloropyridin-2-yl)-4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine
ethyl 4-[(5-phenyl-1,2,4-triazin-3-yl)amino]piperidine-1-carboxylate
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
2-butyl-8-{pyrazolo[1,5-a]pyridine-3-carbonyl}-2,8-diazaspiro[5.5]undecan-3-one
1-[4-(1H-imidazol-1-yl)phenyl]-N-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-amine
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amine
5-(methoxymethyl)-N-({7-[2-(2-methoxyphenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
(2S)-2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-3-(1H-imidazol-4-yl)propanamide
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
N-[3-(1H-imidazol-1-yl)propyl]-4-(piperidin-3-yl)benzamide
5-(2,6-difluorophenoxymethyl)-N-[2-(1,3-thiazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
9-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-5-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazine-1-carbonyl)-4-methyl-1,3-thiazol-2-amine
6-fluoro-2-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)quinolin-4-ol
1-[4-(4-chlorophenoxy)piperidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
N3-[2-(cyclohex-1-en-1-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-N5-(1-methoxypropan-2-yl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-{2-hydroxy-2-[4-(trifluoromethyl)phenyl]ethyl}-1-methyl-1H-1,3-benzodiazole-5-carboxamide
5-cyclopropyl-1-[4-(3-methoxyphenyl)pyrimidin-2-yl]-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
N-benzyl-N-(cyclobutylmethyl)-2-(1H-imidazol-2-yl)benzamide
3-(benzyloxy)-1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)piperidine
N-[1-ethyl-2-(pyridin-3-yl)-7-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1H-1,3-benzodiazol-5-yl]-2-methoxyacetamide
N-{2-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-2-oxoethyl}-N-(3-methylphenyl)methanesulfonamide
4-[(2-methylprop-2-en-1-yl)oxy]-N-[(4-sulfamoylphenyl)methyl]benzamide
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-N-(pyridin-4-ylmethyl)pyridin-2-amine
N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-2,3-dihydro-1H-inden-2-amine