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N-[(3-methoxyphenyl)methyl]-3-[1-(pyridine-3-carbonyl)piperidin-3-yl]propanamide
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
ethyl 4-{3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamido}piperidine-1-carboxylate
(3R,4S)-4-(3-methoxyphenyl)-1-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]pyrrolidin-3-amine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-4-(4-methylphenyl)-5-(pyridin-4-yl)pyrimidin-2-amine
3-[(tert-butylamino)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
N-cyclopropyl-3-[1-(2,5-dimethoxybenzoyl)piperidin-4-yl]propanamide
(3R,4R)-1-(4-ethyl-5-methylpyrimidin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-ol
1-methyl-2-oxo-6-(propan-2-yl)-N-{[4-(trifluoromethyl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
methyl 2-(benzylsulfamoyl)-6-(5-methylpyrazine-2-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 1-(benzyloxy)-2-oxo-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
(1R,5R)-6-(cyclobutylmethyl)-3-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
ethyl 3-[(3-chlorophenyl)methyl]-1-(1H-imidazol-2-ylmethyl)piperidine-3-carboxylate
5-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}thiophene-2-carboxylic acid
N-[(1-cyclopentylpiperidin-3-yl)methyl]-4-oxo-N-[2-(piperidin-1-yl)ethyl]pentanamide
6-[4-(benzyloxy)piperidine-1-carbonyl]quinoline
N,1-dimethyl-N-[2-phenyl-1-(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl)ethyl]-1H-pyrazole-3-carboxamide
N2-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-N4-methylpyrimidine-2,4-diamine
(4aR,7aS)-N,N-dimethyl-6,6-dioxo-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,4-trimethoxybenzamide
(3S,4R)-1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-(3-methylthiophen-2-yl)piperidin-3-ol
{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}dimethylamine
N'-(2-fluoro-5-methylphenyl)-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]butanediamide
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-1-carboxamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-2-(4-phenylpiperidin-1-yl)acetamide
2-amino-3-ethyl-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-(morpholin-4-yl)-3-{1-[(2,3,6-trifluorophenyl)methyl]piperidin-4-yl}propan-1-one
3-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[3-(2,3-dimethylphenoxy)propyl]-N-methylpropanamide
4-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-pyrazole-3-carboxylic acid
1-({5-[(2-fluoro-4-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
1-benzyl-8-(2-phenylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(benzyloxy)-1-(furan-3-carbonyl)piperidine
(1S,5R)-6-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 3-({4-[(2E)-2-methylbut-2-enoyl]-7-oxo-1,4-diazepan-1-yl}methyl)benzoate
4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(naphthalen-1-ylmethyl)morpholine
3-{2-[2-(2-methylphenyl)pyrrolidin-1-yl]-2-oxoethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{7-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-1-[(4-fluorophenyl)methyl]-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
1-benzyl-4-(2,6-dimethylpyridin-4-yl)-1,4-diazepan-6-ol
4-[3-(2-methoxyethyl)-1-propyl-1H-1,2,4-triazol-5-yl]-2,6-dimethylpyridine
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
dimethyl({[(3S,4R)-1-phenylmethanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
5-(2-{[(3-fluorophenyl)methyl]amino}ethyl)-1-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
1-(2-aminoethyl)-N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
2-[(4-chlorophenyl)methyl]-4-{4-[(2-methoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-1,2,4-triazol-1-yl)propan-1-one