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N-[2-(ethylsulfanyl)phenyl]-3-(hydroxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carboxamide
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-(2-chlorophenyl)-3-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-1H-imidazole-5-carboxamide
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
N-(2-{7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
N-cycloheptyl-3-[2-(pyridin-3-yl)piperidin-1-yl]propanamide
N-cyclopropyl-N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)furan-2-carboxamide
3-[(3R,4S)-1-[(4-methoxy-2-methylphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxane-4-carbonyl)piperidine
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
(4aS,8aS)-2-[3-(3-fluorophenyl)benzoyl]-decahydro-2,7-naphthyridin-4a-ol
2,7-dimethyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]pyrazolo[1,5-a]pyrimidine-5-carboxamide
(1R,5R)-6-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-{4-[4-(3-hydroxyazetidine-1-carbonyl)phenoxy]piperidin-1-yl}-3-methoxypropan-1-one
N-butyl-4-methyl-3-phenyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
N-(1-{7-[(3-ethoxy-4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
8-(2-methylpyridin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 2-(4-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2-oxopiperazin-1-yl)acetate
1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazole
2-{[(cyclopropylmethyl)amino]methyl}-6-methylquinolin-4-ol
2-(morpholin-2-yl)-1-[4-(quinazolin-4-yl)piperazin-1-yl]ethan-1-one
[4-({1-[(3-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-({1-[6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-3-yl}methyl)acetamide
2-(2-hydroxyethyl)-9-[5-(propan-2-yl)pyrimidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
8-methoxy-2-{[2-(3-methoxypropyl)piperidin-1-yl]methyl}quinoline
3-(1-methyl-1H-pyrazol-5-yl)-1-[4-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
2-(4-{[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]methyl}phenoxy)-1-(morpholin-4-yl)ethan-1-one
4-chloro-3-{3-[(1-methylpiperidin-4-yl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}-1H-pyrazol-5-amine
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-[2-(piperidin-1-yl)ethyl]benzamide
4-pentanamido-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]benzamide
1-[2-methyl-7-(thiophen-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperidin-3-ol
methyl 6-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]amino}-1,2,3,4-tetrahydroquinoline-1-carboxylate
N-(1-{1-[(2-chloro-4-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
4-{5-[(cyclohexylmethyl)sulfanyl]-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl}-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-[(2-methylphenyl)methyl]-N-(prop-2-en-1-yl)acetamide
4-(2,6-dimethylpyridin-3-yl)-2-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine
4-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
1-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
3-[7-(2-phenylacetyl)-2,3-dihydro-1,4-benzodioxin-6-yl]propanamide
(1R,5S)-3-{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 3-({1-methyl-3-[(thiophen-2-ylmethyl)carbamoyl]-4,5,6,7-tetrahydro-1H-indazol-5-yl}amino)propanoate
3-methoxy-2,2-dimethyl-1-[3-(pyridin-2-yl)azetidin-1-yl]propan-1-one
5-(3-acetylphenoxymethyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]-1,2-oxazole-3-carboxamide
({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(propyl)(pyridin-3-ylmethyl)amine
3-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}ethyl]methylamine
1-(1-benzothiophene-2-carbonyl)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)piperidin-3-amine
[(3R,4R)-1-[(7-chloro-3-methyl-1H-indol-2-yl)methyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol