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4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-methylpiperazin-2-yl}methanol
6-[(1H-indol-6-ylmethyl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-methyloxane-2-carboxamide
2-[(3-{[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]carbamoyl}phenyl)amino]acetic acid
(3aR,6aR)-2-acetyl-5-{[2-(butylsulfanyl)pyrimidin-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(furan-2-yl)-2-oxoacetamide
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
1-(2-{7-[(3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)piperidin-2-one
N-(1-{5-[(cyclohexylmethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}-2-phenylethyl)-2,4-dimethoxybenzamide
5-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-[(2-fluorophenyl)methyl]-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
2-(dimethylamino)-1-[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]-2-(3-methylphenyl)ethan-1-one
1-(4-{[3-(hydroxymethyl)-3-[(3-methoxyphenyl)methyl]piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
3-{[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]sulfamoyl}-N-(oxolan-3-yl)benzamide
6-(2-chlorophenyl)-N-methyl-N-(oxan-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]benzamide
2-{4-[(5-ethylfuran-2-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
1-benzyl-5-(2,3-dimethoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
1-[1-({1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
5-(5-cyclopropyl-1,3-oxazol-4-yl)-3-(diphenylmethyl)-1,2,4-oxadiazole
2,2-dimethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)oxane-4-carboxamide
9-(cyclopropylmethyl)-4-[(4-fluoro-2-methylphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
5-(2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
1-[5-({[(1-ethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-ethyl-N-(oxolan-2-ylmethyl)acetamide
N-cyclopropyl-6-(2-methylphenyl)-N-(oxan-4-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(3S,4R)-1-[(6-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-[(4aR,8aS)-6-methanesulfonyl-decahydro-1,6-naphthyridin-1-yl]-2-(3,4,5-trifluorophenyl)ethan-1-one
4-({2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl)amino)-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-N-(1-methyl-1H-pyrazol-3-yl)acetamide
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(2-ethoxyphenyl)piperazine
2-[2-(1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
3-[(4-fluorophenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)propanamide
2-(4-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
3-{2-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-oxoethyl}-4-(3-methylbutyl)piperazin-2-one
2-methyl-5-{[3-(3-methylpiperidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}pyridine
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(3-methylpyridin-2-yl)methyl]piperazine
4-{1-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-1H-1,2,3-triazol-4-yl}-1-(propan-2-yl)piperidine
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-4-methyl-1H-imidazole-5-carboxamide
2-(1H-pyrazol-1-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N,5-dimethyl-N-(1,3-thiazol-2-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
5-[(2,3-dihydro-1H-inden-2-yl)amino]-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-{[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]carbamoyl}pyrrolidine-2-carboxylic acid
1-methyl-4-{1-[2-(3-methylthiophen-2-yl)ethyl]-1H-imidazol-2-yl}piperidine
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-[2-(3-methylpyridin-2-yl)ethyl]benzamide
2-[(4-{2-[2-(pyridin-2-yl)ethyl]piperidine-1-carbonyl}phenyl)sulfanyl]ethan-1-ol
N-[2-(dimethylsulfamoyl)ethyl]-3-(piperidin-3-yl)benzamide