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(3S,4S)-4-methoxy-N-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-amine
1-[2-(4-methoxyphenyl)ethyl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]-6-oxopiperidine-3-carboxamide
2-(4-chlorophenyl)-N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)acetamide
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(3-methoxyphenyl)-1-[1-(2-phenoxyacetyl)piperidin-4-yl]ethyl]-N,1-dimethyl-1H-pyrazole-3-carboxamide
1-[(3-methoxyphenyl)methyl]-N-[(5-methylfuran-2-yl)methyl]-6-oxopiperidine-3-carboxamide
N-(4-{1-[1-(furan-2-carbonyl)piperidin-3-yl]-1H-1,2,3-triazol-4-yl}phenyl)acetamide
2-[1-(3-phenylpropyl)-4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
4-{4-[(4-ethylphenyl)methyl]piperazin-1-yl}-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
5-[4-(5-chloro-2-methylphenyl)piperazin-1-yl]-1-ethyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
N-[2-(cyclohexylsulfanyl)ethyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
8-(4-aminocyclohexyl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
5-({1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}carbamoyl)-1H-imidazole-4-carboxylic acid
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-4-ethenylbenzamide
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-2-[N-(3-methylphenyl)methanesulfonamido]acetamide
5-(2-fluorophenoxymethyl)-N-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide
1-(1-{1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
9-methoxy-3-(2-phenylpropyl)-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-4-(3,5-dimethyl-1H-pyrazol-1-yl)butan-1-one
1'-[2-(3-hydroxyphenyl)acetyl]-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-[(1,2-oxazol-3-ylmethyl)sulfamoyl]benzamide
3-(2,3-dihydroxypropyl)-1-(5-fluoro-2-methoxyphenyl)urea
(1S,5R)-6-(cyclopropylmethyl)-3-[2-(3-methylphenyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-fluoropiperidine
4-[4-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)phenyl]-2-methylbutan-2-ol
(3S,4R)-N,N-dimethyl-1-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-4-propylpyrrolidin-3-amine
(2R,3S,6R)-5-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-propanamido-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
3-({3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}methoxy)pyridine
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
9-[3-(1H-pyrazol-1-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-(cyclopropylmethyl)-5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{5-[2-(azocan-1-yl)ethyl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
7-[5-(hydroxymethyl)furan-2-carbonyl]-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[2-(3-methoxyphenyl)ethyl]-4-{4-[4-(3-methoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide
3-{[1-(3,4-dihydro-2H-1,5-benzodioxepin-7-yl)ethyl]amino}-N-(furan-2-ylmethyl)propanamide
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
N4-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyrimidine-2,4-diamine
N-(3-ethoxypropyl)-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
4-[4-(4-chlorophenyl)-5-methyl-1H-imidazol-2-yl]-1-(2-methylpropyl)pyrrolidin-2-one
ethyl 5-(5-acetylthiophene-3-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
5-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methyl-1H-1,3-benzodiazole
1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-3-(2-methoxyphenoxy)azetidine
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
3,7-dimethyl-2-({4-[2-(piperidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)-1H-indole
2-(1H-indazol-3-yl)-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}acetamide