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2-({2-[(2,5-dimethylphenyl)carbamoyl]ethyl}amino)-N-(1,3-thiazol-2-yl)propanamide
(3S,4S)-4-cyclopropyl-1-(2-methoxy-5-methylbenzenesulfonyl)pyrrolidine-3-carboxylic acid
4-benzyl-3-ethyl-1-(1-methyl-1H-imidazole-5-carbonyl)-1,4-diazepan-5-one
4-{6-[3-(pyridin-3-yl)azetidin-1-yl]pyrazine-2-carbonyl}morpholine
4-(3-{[(1-methoxypropan-2-yl)amino]methyl}phenyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(2,3-dihydro-1H-inden-5-yl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
N-[1-(4-methyl-1H-imidazol-2-yl)propyl]-4-(trifluoromethyl)benzamide
6-methyl-2-{[4-(2-methyl-5-propylpyrimidin-4-yl)piperazin-1-yl]methyl}pyridin-3-ol
(1R,5R)-N,N-dimethyl-6-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(1-methyl-1H-imidazol-2-yl)methyl]-1,4-diazepane
4-({2-[1-(5-phenyl-1,2,4-oxadiazol-3-yl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}[(2-methylphenyl)methyl](pyridin-4-ylmethyl)amine
3,6-dimethyl-N-[2-(quinolin-8-yloxy)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-(furan-3-ylmethyl)-3-(2-{8-methoxy-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}-2-oxoethyl)piperazin-2-one
2-[4-(4-cyclopentylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-4-(3-methoxyphenyl)pyrimidine
3-(methoxymethyl)-5-[2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethyl]-1,2,4-oxadiazole
N-ethyl-1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-3-carboxamide
3-(4-methyl-4H-1,2,4-triazol-3-yl)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]propan-1-one
3-(but-2-yn-1-yl)-5-[1-(3-chloro-2-fluorobenzoyl)piperidin-4-yl]-5-(2-phenylethyl)imidazolidine-2,4-dione
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(1,2-oxazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
(4aR,8aR)-7-(2,5-dimethylfuran-3-carbonyl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
1-[(2-chlorophenyl)methyl]-N-methyl-N-[2-methyl-3-(pyrrolidin-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
N-(2-fluoro-5-methylphenyl)-3-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]propanamide
1-[(3R,4S)-3-[(2-methylpyrimidin-4-yl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
4-(1H-indol-3-ylmethyl)-1-[(4-methoxyphenyl)methyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
methyl (2S)-2-[(1-{4-[(dimethylsulfamoyl)amino]phenyl}piperidin-4-yl)amino]-2-phenylacetate
3-[2-(dimethylamino)ethyl]-1-ethyl-8-{[4-(methylsulfanyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
N-benzyl-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N,N-dimethyl-3-[4-(thiophen-2-yl)butanamido]azepane-1-carboxamide
2-(dimethylamino)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-(3-methylphenyl)acetamide
8-methoxy-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[1-(2-methyl-1,3-benzothiazol-6-yl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
2-(dimethylamino)-N-[2-(ethylsulfanyl)ethyl]-2-(3-fluorophenyl)acetamide
(3S,7S,8aS)-7-{[(2-fluorophenyl)methyl]amino}-3-(hydroxymethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
N-[(3R,4S)-1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
ethyl 4-[4-(4-{[3-(pyridin-3-yl)propyl]amino}piperidin-1-yl)benzoyl]piperazine-1-carboxylate
3-ethyl-N-[(1R,2R)-2-hydroxycyclohexyl]-1H-indole-2-carboxamide
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-ethyl-5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]furan-2-carboxamide
({2-methoxy-5-[1-(3-methylbutan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}methyl)dimethylamine
1-(1-methyl-1H-pyrazole-3-carbonyl)-4-(4-methylphenoxy)piperidine
4-cyclopropanecarbonyl-7-(phenoxathiin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
N,2,4-trimethyl-N-[1-(pyridin-3-yl)pentyl]-1,3-thiazole-5-carboxamide
N,5-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1,2-oxazole-3-carboxamide
3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(2-phenylethyl)propanamide
1-(1H-indole-6-carbonyl)-N,N-dimethylazepan-4-amine
N-cyclohexyl-4-{[1-(morpholin-4-yl)propan-2-yl]amino}piperidine-1-carboxamide