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N-{1-[(2-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-(4-methylphenoxy)acetamide
1-{[4-(1-ethyl-1H-1,2,4-triazol-5-yl)phenyl]methyl}-1H-1,2,3,4-tetrazole
3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}-1-phenylpyrrolidin-2-one
1-(5-methylpyridine-3-carbonyl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
8-(3-aminopropanoyl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{3-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}methanesulfonamide
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(quinolin-5-ylmethyl)piperidine-2-carboxamide
N5-cyclooctyl-N3-methyl-4-oxo-1-(oxolan-2-ylmethyl)-N3-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(2-fluoro-5-methoxyphenyl)-6-(piperidine-1-carbonyl)pyrazine
1-[3-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)propyl]piperidin-3-ol
N-{[8-(pyridin-4-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
4-hydroxy-2-methyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrimidine-5-carboxamide
N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}cyclohex-3-ene-1-carboxamide
N-methyl-5-(phenoxymethyl)-N-(3-phenylpropyl)-1H-pyrazole-3-carboxamide
1-cyclohexyl-4-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
N-(oxolan-3-yl)-1-[4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)phenyl]piperidin-4-amine
2-[methyl({5-[(3-phenylpiperidin-1-yl)methyl]pyrimidin-2-yl})amino]acetic acid
N-{[4-(aminomethyl)phenyl]methyl}-2-(4,6-dimethyl-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
N-(9H-fluoren-9-yl)morpholine-2-carboxamide
N-[3-(furan-2-yl)-3-phenylpropyl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(1-methylpyrrolidin-2-yl)ethyl]amine
N-({5-[(4-chloro-2-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
4-(4-chlorophenyl)-1-[3-(2-phenylpropyl)-1,2-oxazole-5-carbonyl]piperidin-4-ol
(2S)-2-hydroxy-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]formamido}butanoic acid
N-(3,4-difluorophenyl)-2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-5-ethyl-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
3-(but-2-yn-1-yl)-5-(3-phenylpropyl)-5-{1-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]piperidin-4-yl}imidazolidine-2,4-dione
2-{[(1-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]sulfanyl}pyridine
5-{3-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-3-oxopropyl}-5-(thiophen-3-ylmethyl)pyrrolidin-2-one
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-2-oxo-2-(2-phenylindolizin-3-yl)acetamide
4-(4-benzyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-butylpiperidine-1-carboxamide
N-[(3S,4R)-1-{2-[(2-fluorophenyl)amino]acetyl}-4-propylpyrrolidin-3-yl]acetamide
3-(oxolan-3-yl)-5-[2-(thiophen-2-yl)ethyl]-1,2,4-oxadiazole
4-{3-[2-(3-chlorophenyl)-1H-imidazol-1-yl]-4-methoxyphenyl}-4H-1,2,4-triazole
4-(2-oxo-2-{spiro[azepane-4,2'-chromene]-1-yl}ethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
5-{1-[(2E)-3-(2-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
1-(4-ethenylbenzoyl)-4-(piperidine-1-carbonyl)piperidine
5-[2-(morpholine-4-carbonyl)piperazine-1-carbonyl]quinoxaline
N-(cyclopropylmethyl)-5-methyl-4-[(oxolan-2-ylmethyl)amino]-N-propylthieno[2,3-d]pyrimidine-6-carboxamide
1-(4-methoxybenzoyl)-4-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
(2H-1,3-benzodioxol-5-ylmethyl)[3-(methylsulfanyl)butyl](pyridin-3-ylmethyl)amine
4,6-dimethyl-3-{4-[3-oxo-3-(4-phenylpiperazin-1-yl)propyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[2-(oxan-2-yl)ethyl]propanamide
3-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)amino}methyl)piperidin-3-ol
methyl 3-[(2-methoxyphenyl)methyl]-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(2-methoxyphenyl)-N-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-1H-pyrazole-4-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(furan-2-yl)-N-[2-(4-methylpiperazin-1-yl)phenyl]-1H-pyrazole-4-carboxamide
methyl (2S,3S)-2-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}formamido)-3-methylpentanoate
3-[(2,3-dimethoxyphenyl)methyl]-9-methoxy-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide