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3-(3,5-dimethylphenyl)-1-[4-(pyridin-4-yloxy)piperidin-1-yl]propan-1-one
(2R)-2-cyclohexyl-N-[2-(4,5-dimethyl-1H-imidazol-1-yl)ethyl]-2-hydroxyacetamide
N-{[5-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-3-yl]methyl}-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-[(3R,4R)-1-(2-aminopyrimidin-4-yl)-3-hydroxypiperidin-4-yl]-N-ethyl-2,3-difluorobenzamide
N-[4-(2,5-dimethylphenyl)-8-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-methoxyacetamide
N-(3-{4-[methyl({[4-(trifluoromethyl)phenyl]methyl})amino]piperidin-1-yl}phenyl)pyridine-4-carboxamide
methyl 3-[(3S,4R)-1-[(2,4-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]propanoate
(4S,4aS,8aS)-1-(4-methyl-1,3-thiazole-5-carbonyl)-4-phenyl-decahydroquinolin-4-ol
N-[(5-methylfuran-2-yl)methyl]-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
3-(2-methoxyethyl)-8-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2,3-dimethyl-N-(4-pentanamidophenyl)-1H-indole-5-carboxamide
2-(4-fluorophenyl)-1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperidine
methyl 2-(azocane-1-sulfonyl)-6-[3-(methylsulfanyl)propanoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-cyclopentyl-4-({[4-(pyridin-3-yl)pyrimidin-2-yl]amino}methyl)pyrrolidin-2-one
5-[(2-chlorophenyl)methyl]-5-(piperidin-4-yl)-3-(1,3-thiazol-5-ylmethyl)imidazolidine-2,4-dione
N-(3,3-diphenylpropyl)-4-[4-(2-methoxyacetamido)-1H-pyrazol-1-yl]benzamide
N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]pyrazine-2-carboxamide
N-({7-[(3-hydroxy-4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
5-cyclopentyl-1-{[1-(methoxymethyl)cyclopropyl]methyl}-4-phenyl-1H-imidazole
N-({1-butyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}methyl)methanesulfonamide
methyl (1S,3S,3aR,6aS)-1-(hydroxymethyl)-3-(4-methoxy-2-methylphenyl)-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-cyclobutyl-5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-amine
3-(4-methyl-1,3-thiazol-5-yl)-N-[(3-methyl-1-benzofuran-2-yl)methyl]propanamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]methylamine
N-butyl-1-cyclohexyl-4-oxo-5-(4-phenylpiperazine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-[4-(pyrazin-2-yl)piperazin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
methyl 3-{[4-(methoxycarbonyl)phenyl]methyl}-7-oxo-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}piperidin-2-one
N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]ethane-1-sulfonamide
7-methoxy-3-({[1-(naphthalen-1-yl)ethyl]amino}methyl)-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-2-one
2-{1-[(3-methoxyphenyl)methyl]-4-[(3-methylquinoxalin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
2-chloro-N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
5-[(2-chlorophenyl)methyl]-5-{1-[2-(2-methoxyphenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
2-(3-methylbut-2-en-1-yl)-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
8-(5-methyl-1,3-oxazole-4-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-3-{1-[4-(4-methylpiperazin-1-yl)benzoyl]piperidin-4-yl}propanamide
4-(1-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-4-yl}ethyl)morpholine
2-[2-(1-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}piperidin-2-yl)ethyl]pyridine
4-amino-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}pyridine-2-carboxamide
3-[({[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}amino)methyl]piperidin-3-ol
1-propanoyl-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2-(aminomethyl)-N-(3-carbamoyl-2-methylphenyl)piperidine-1-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-3-ol
7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(pyrrolidine-1-carbonyl)piperazine
3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1-[2-(morpholin-4-ylmethyl)phenyl]urea
methyl 2-(azocane-1-sulfonyl)-6-(1,3-thiazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-3-(methylsulfanyl)-N-(oxolan-2-ylmethyl)propanamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide